Hindered N-oxide esters of rapamycin

Details Hindered N-oxide esters of rapamycin Hindered N-oxide esters of rapamycin

1995-05-24

1996-04-16

Bond, Robert T.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Phosphorus containing other than solely as part of an...

540456, A61K 31395, C07D49516

Patent

active

055082904

ABSTRACT:
A compound of the structure ##STR1## wherein R and R.sup.1 are each, independently, ##STR2## or hydrogen; R.sup.2 and R.sup.3 are each, independently, alkyl, arylalkyl , or R.sup.2 and R.sup.3 may be taken together to form a cycloalkyl ring;

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