Hexahydro-1-arylspiro(3H-oxazolo(3,4-A)pyridine-3,4'-piperidene)

Drug – bio-affecting and body treating compositions – Antigen – epitope – or other immunospecific immunoeffector – Parasitic organism or component thereof or substance...

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546 17, 546 19, 546241, 546242, 546216, C07D49820, A61K 31445

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active

042606233

ABSTRACT:
Compounds of the formula ##STR1## where R.sub.1 is hydrogen, lower alkyl containing one to three carbon atoms, cycloalkyl lower alkyl containing four to seven carbon atoms, or benzyl; and R.sub.2 is hydrogen, halogen, alkoxy containing one to three carbon atoms, trifluoromethyl; and pharmaceutically acceptable acid addition salts thereof are useful as anti-depressants.

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Novel Tetracycic Spiropiperidines and Related Compounds as Potential Psychotropic Agents, L. L. Martin et al., Am. Chem. Soc., Div. of Med. Chem., 178th National Meeting, Sep. 10 to 13, 1979, Washington, D.C.
Arya et al., "Indian J. Chem.", Section B (1976), vol. 14B, No. 10, pp. 777-779.
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