Heteropolycyclic inhibitors of protein kinases

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Reexamination Certificate

active

10310600

ABSTRACT:
A method of inhibiting tumor growth is provided, comprising administering an effective dose of a compound of the formulawherein, independently at each occurrence,w is C or N, v and x are N with H substitution as needed to fulfill open valence sites;y and z are selected from N and C, with H substitution as needed to fulfill open valence sites, with the proviso that each of w, v, x, y and z is not simultaneously C;the ring formed from v, w, x, y and z may be saturated or unsaturated; andR1, R2, R3and R4are selected from hydrogen, alkyl, aryl, alkaryl, aralkyl, heteroalkyl, and heteroaryl; wherein any adjacent two of R1, R2, R3and R4may join together to form a 5, 6 or 7-membered carbocyclic ring or a 5, 6 or 7-membered heterocyclic ring containing at least one atom selected from nitrogen, oxygen and sulfur.

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patent: 01/79209 (2001-10-01), None
Kane et al. (1999), “Induction of NF-κB by the Akt/PKB Kinase,”Current Biology, vol. 9:601-604.
Junek et al.,Syntheses with nitriles XLV 2-(1, 3-Dioxo-2-indanylidene)benzimidazoline-and isomer of indigo, Inst. Org. Chem., 1977, 2276-82, 110(6), Univ. Graz, Graz, Austria.

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