Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-01-17
1996-12-10
Chang, Ceila
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514183, 514200, 514212, 5142315, 5142338, 5142345, 5142352, 5142355, 5142358, 5142368, 5142372, 514252, 514256, 514258, 514266, 514303, 514314, 514316, 514318, 514319, 514321, 540200, 540354, 540480, 540483, 540544, 540553, 540597, 540600, 540603, 544124, 544127, 544128, 544129, 544130, 544133, 544135, 544137, 544139, 544141, 544238, 544242, 544277, 544283, 544336, 546118, 546152, 546190, 546193, 546198, 546208, 546209, 546210, 546211, 546212, 546214, A61K 31445, A61K 3140, C07D40112, C07D20709, C07D211;280
Patent
active
055831460
ABSTRACT:
Heterocyclic thrombin inhibitors are provided which have the structure ##STR1## wherein n, R, R.sup.1, R.sup.2, R.sup.3, G, G.sub.x, R.sup.6', Ra, Xa, R.sup.6, Rb, R.sub.3, p, Q, A and R.sup.4 are as defined herein.
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Das Jagabandhu
Hall Steven E.
Han Wen-Ching
Kimball Spencer D.
Lau Wan F.
Bristol--Myers Squibb Company
Chang Ceila
Rodney Burton
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