Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1997-08-26
2000-12-26
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
540544, A61K 3155, C07D 28106
Patent
active
061660051
ABSTRACT:
The invention provides compounds of formula ##STR1## as described in the claims, or an optical isomer, diastereomer or enantiomer thereof, or a pharmaceutically-acceptable salt, or biohydrolyzable amide, ester, or imide thereof are useful as inhibitors of metalloproteases. Also disclosed are pharmaceutical compositions and methods of treating diseases, disorders and conditions characterized by metalloprotease activity using these compounds or the pharmaceutical compositions containing them.
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Almstead Neil Gregory
Cheng Menyan
De Biswanath
Matthews Randall Stryker
Natchus Michael George
Roof Carl J.
Shah Mukund J.
Sripada Pavanaram K
The Procter & Gamble & Company
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