Heterocyclic hydrazones for use as anti-cancer agents

Details Heterocyclic hydrazones for use as anti-cancer agents Heterocyclic hydrazones for use as anti-cancer agents

2006-09-26

2006-09-26

Wilson, James O. (Department: 1624)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C548S302700, C548S302400

Reexamination Certificate

active

07112680

ABSTRACT:
The invention relates to novel 2-benzimidazolyl-, 2-benzoxazolyl- and 2-benzothiazolyl hydrazones that are derived from 2-formylpyridine, 2-acylpyridines, acetyldiazines and acetyl(iso)quinolines. The invention also relates to a novel method for producing 2-benzimidazolyl-, 2-benzoxazolyl- and 2-benzothiazolyl hydrazones and to their use as useful anti-cancer therapeutic agents. The novel compounds are also active against multidrug-resistant cancer cells.

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