Organic compounds -- part of the class 532-570 series – Organic compounds – Nitrogen attached directly or indirectly to the purine ring...
Patent
1994-03-28
1996-09-17
Gibson, Sharon
Organic compounds -- part of the class 532-570 series
Organic compounds
Nitrogen attached directly or indirectly to the purine ring...
544364, 544365, C07D40100
Patent
active
055569773
ABSTRACT:
Compounds of formula I ##STR1## and metabolically labile esters and amides thereof, and pharmaceutically acceptable salts thereof, in which R.sup.13, M.sup.2, X.sup.1, Z.sup.1, Z.sup.1a, X.sup.2 and A.sup.1 have the meanings given in the specification. The compounds are useful as inhibitors of the binding of fibrinogen to glycoprotein IIb/IIIa. Intermediates are also disclosed.
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Brewster Andrew G.
Caulkett Peter W. R.
Faull Alan W.
Mills Sturat D.
Pearce Robert J.
Gibson Sharon
Kilby Scalzo Catherine
Zeneca Limited
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