Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Phosphorus containing other than solely as part of an...
Reexamination Certificate
2007-06-26
2007-06-26
Berch, Mark L. (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Phosphorus containing other than solely as part of an...
C514S234200, C514S218000, C514S212020, C514S263200, C514S263220, C540S575000, C544S244000, C544S118000, C544S061000, C544S269000, C544S271000, C544S272000, C544S231000
Reexamination Certificate
active
10621302
ABSTRACT:
The present invention relates to therapeutically active and selective inhibitors of the enzyme DPP-IV, which are of formula Iwherein each n is one or two independently and R1, R2, R3, R6, R7, R9, and R10are defined herein. The present invention also relates to pharmaceutical compositions comprising the compounds of formula I and the use of the compounds for treating diseases that are associated with proteins that are subject to inactivation by DPP-IV, such as type-2 diabetes and obesity.
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Christiansen Lise Brown
Kanstrup Anders Bendtz
Kristiansen Marit
Lundbeck Jane Marie
Sams Christian K.
Berch Mark L.
Bork Richard W.
Novo Nordisk A S
Wilk-Orescan Rosemarie R.
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