Heterocyclic compounds

Details Heterocyclic compounds Heterocyclic compounds

1998-12-14

2000-04-11

Davis, Zinna Northington

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

546203, 540587, 514325, A61K 3155, A61K 31435, C07D21106, C07D22318

Patent

active

060488565

ABSTRACT:
The present invention relates to novel N-substituted azaheterocyclic compounds of the formula ##STR1## wherein X, Y, R.sup.1, R.sup.1a, R.sup.2, R.sup.2a, R.sup.12, R.sup.13, A, r and s are as defined in the detailed part of the present description, or salts thereof, to methods for their preparation, to compositions containing them, and to their use for the clinical treatment of painful, hyperalgesic and/or inflammatory conditions in which C-fibers play a pathophysiological role by eliciting neurogenic pain or inflammation. These compounds are also useful for treating indications caused by or related to the secretion and circulation of insulin antagonizing peptides, e.g., non-insulin-dependent diabetes mellitus (NIDDM) and ageing-associated obesity.

REFERENCES:
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Chemical Abstract, vol. 66, No. 13, p. 5247 (Mar. 27, 1967).
Chemical Abstract, vol. 59, No. 8, abstract No. 8750 (Oct. 14, 1963).
Chemical Abstract, vol. 127, No. 19, p. 633 (Nov. 10, 1997) Miyamoto, et al.
Chemical Abstract, vol. 72, No. 1 p. 308 (Jan. 5, 1970).
Chemical Abstract, vol. 123, No. 23, p. 908 (Dec. 4, 1995).

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