Heterocyclic antiviral compounds

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Phosphorus containing other than solely as part of an...

Reexamination Certificate

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Details

C514S248000, C544S232000, C544S236000

Reexamination Certificate

active

08063028

ABSTRACT:
Compounds of formula I, wherein R1, R2, R3, X1, X2and Ar, are as defined herein or pharmaceutically acceptable salts thereof, inhibit HIV-1 reverse transcriptase and afford a method for prevention and treatment of HIV-1 infections and the treatment of AIDS and/or ARC. The present invention also relates to compositions containing compounds of formula I useful for the prevention and treatment of HIV-1 infections and the treatment of AIDS and/or ARC.

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Chan, J. H., et. al. “Novel Bensophenones as Non-Nucleoside Reverse Transcriptase Inhibitors of HIV-1,”Journal of Medicinal Chemistry, 2004, vol. 47, pp. 1175-1182.
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