Heterocycle-substituted benzimidazole derivative

Details Heterocycle-substituted benzimidazole derivative Heterocycle-substituted benzimidazole derivative

2011-08-09

2011-08-09

Saeed, Kamal (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C514S338000

Reexamination Certificate

active

07994331

ABSTRACT:
A compound represented by the formula (I) or a pharmaceutically acceptable salt thereof: (I) wherein X1to X4independently represent a carbon atom or the like; the ring A represents a 5- to 6-membered heteroaryl having 1 to 4 heteroatoms independently selected from the group consisting of a nitrogen atom, a sulfur atom and an oxygen atom; X5represents an oxygen atom or the like; X represents a carbon atom or the like; Het represents a 5- or 6-membered aliphatic heterocycle; R1represents an aryl or the like; R2represents a formyl group or the like; and R3represents a —C1-6alkyl or the like. The compound or salt has a glucokinase activation effect and is useful as a therapeutic agent for diabetes.

REFERENCES:
patent: 6187805 (2001-02-01), Pineiro et al.
patent: 6316468 (2001-11-01), Maxey et al.
patent: 6433188 (2002-08-01), Corbett et al.
patent: 6441184 (2002-08-01), Corbett et al.
patent: 6448399 (2002-09-01), Corbett et al.
patent: 6518273 (2003-02-01), Chapman et al.
patent: 6545155 (2003-04-01), Corbett et al.
patent: 6723725 (2004-04-01), Bottcher et al.
patent: 7253286 (2007-08-01), Funahashi et al.
patent: 7301036 (2007-11-01), Parmee et al.
patent: 2002/0103199 (2002-08-01), Corbett et al.
patent: 2002/0103241 (2002-08-01), Corbett et al.
patent: 2002/0107396 (2002-08-01), Corbett et al.
patent: 2002/0111372 (2002-08-01), Corbett et al.
patent: 2004/0053908 (2004-03-01), Funahashi et al.
patent: 2005/0153980 (2005-07-01), Schadt et al.
patent: 2006/0063811 (2006-03-01), Hoelzemann et al.
patent: 2006/0160824 (2006-07-01), Heinrich et al.
patent: 2006/0160832 (2006-07-01), Funahashi et al.
patent: 2006/0247259 (2006-11-01), Funahashi et al.
patent: 2007/0093544 (2007-04-01), Parmee et al.
patent: 2007/0099933 (2007-05-01), Heinrich et al.
patent: 2007/0105930 (2007-05-01), Parmee et al.
patent: 2008/0070928 (2008-03-01), Nonoshita et al.
patent: 2008/0125429 (2008-05-01), Hashimoto et al.
patent: 2586056 (2006-05-01), None
patent: 1 810 969 (2007-07-01), None
patent: 2004-67629 (2004-03-01), None
patent: 2004-517087 (2004-06-01), None
patent: WO 02/32872 (2002-04-01), None
patent: WO 02/39989 (2002-05-01), None
patent: WO 2003/087086 (2003-10-01), None
patent: WO 2004/014300 (2004-02-01), None
patent: WO 2004/026248 (2004-04-01), None
patent: WO 2004/100875 (2004-11-01), None
patent: WO 2004/113325 (2004-12-01), None
patent: WO 2004/113326 (2004-12-01), None
patent: WO 2005/054193 (2005-06-01), None
patent: WO 2005/063738 (2005-07-01), None
patent: WO 2005/065680 (2005-07-01), None
patent: WO 2006/014262 (2006-02-01), None
patent: WO 2006/049304 (2006-05-01), None
patent: WO 2006/074789 (2006-07-01), None
patent: WO 2007/019675 (2007-02-01), None
patent: WO 2007/021629 (2007-02-01), None
patent: WO 2007/061763 (2007-05-01), None
patent: WO 2007/121578 (2007-11-01), None

Affiliated with

Also associated with

Rating

Heterocycle-substituted benzimidazole derivative does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Heterocycle-substituted benzimidazole derivative, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Heterocycle-substituted benzimidazole derivative will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2684489