Heteroaryl derivatives and their use as medicaments

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C544S333000, C544S361000, C514S256000

Reexamination Certificate

active

06936615

ABSTRACT:
The invention relates to novel quinoline derivatives of the formula 1, to their preparation and to their use as medicaments, in particular for treating tumors.

REFERENCES:
patent: 4656174 (1987-04-01), Campbell et al.
patent: 4937246 (1990-06-01), Sugihara et al.
patent: 5432175 (1995-07-01), Dyke et al.
patent: 5804588 (1998-09-01), Dyke et al.
patent: 5861395 (1999-01-01), Taveras et al.
patent: 6706722 (2004-03-01), Emig et al.
patent: 0112 776 (1984-07-01), None
patent: 0 831 090 (1998-03-01), None
patent: WO 95/00497 (1995-01-01), None
patent: WO 97/44329 (1997-11-01), None
patent: WO 98/00402 (1998-01-01), None
patent: WO 99/02520 (1999-01-01), None
patent: WO 99/16751 (1999-04-01), None
patent: WO 00/12074 (2000-03-01), None
patent: WO 00/51614 (2000-09-01), None
Chemical Abstract, abstract of WO 99/02520.
Examination Report of the corresponding Chinese Patent Application.
Todd R. Elworthy, Anthony P.D.W. Ford, Gary W. Bantle, et al., N-Arylpiperazinyl-N′-propylamino Derivatives of Heteroaryl Amides as Functional Uroselective a1-Adrenoceptor Antagaonists, J. Med. Chem. 1997, 40, 2674-2687.
Arthur G. Taveras, Jeff Deskus, Jianping Chao, Cynthia J. Caccaro, et al., Identification of Pharmacokinetically Stable 3, 10-Dibromo-8-chlorobenzocycloheptapyridine Farnesyl Protein Transferase Inhibitors with Potent Enzyme and Cellular Activities, J. Med Chem. 1999, 42, 2651-2661.
El-Sebai A. Ibrahim, I. Chaaban and S. M. El-Khawass, Synthesis of Some Quinoline Derivatives of Potential Antiamebic Activity, Pharmazie 32, H. 3 (1977), 155-156.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Heteroaryl derivatives and their use as medicaments does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Heteroaryl derivatives and their use as medicaments, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Heteroaryl derivatives and their use as medicaments will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-3449308

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.