Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2006-02-07
2006-02-07
Raymond, Richard (Department: 1623)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C546S001000, C514S352000, C514S218000, C514S252120, C514S254100, C540S575000, C564S163000, C564S164000, C544S400000, C544S374000
Reexamination Certificate
active
06995269
ABSTRACT:
Compounds of formula IIA and IIB are novel guanidine compoundswhere the variables R1through R10have the values set forth herein. Such compounds have use in treating diseases such as obesity and type II diabetes, and may be provided as pharmaceutical formulations in conjunction with a pharmaceutically acceptable carrier.
REFERENCES:
patent: 3177218 (1965-04-01), Brown
patent: 4128643 (1978-12-01), Merkel et al.
patent: 4287341 (1981-09-01), Hess et al.
patent: 4496571 (1985-01-01), Yellin et al.
patent: 4732916 (1988-03-01), Satoh et al.
patent: 4748165 (1988-05-01), Jones et al.
patent: 4874864 (1989-10-01), Schnur et al.
patent: 4948891 (1990-08-01), Schnur et al.
patent: 4948901 (1990-08-01), Schnur et al.
patent: 5086057 (1992-02-01), Sasagawa
patent: 5124328 (1992-06-01), Fisher et al.
patent: 5352704 (1994-10-01), Okuyama et al.
patent: 5362902 (1994-11-01), Barnish et al.
patent: 5547966 (1996-08-01), Atwal et al.
patent: 5637439 (1997-06-01), Kaneko et al.
patent: 5750573 (1998-05-01), Bianchi et al.
patent: 5885985 (1999-03-01), Macdonald et al.
patent: 5889025 (1999-03-01), Lohray et al.
patent: 5952381 (1999-09-01), Chen et al.
patent: 5962530 (1999-10-01), Engel et al.
patent: 6020349 (2000-02-01), Ankersen et al.
patent: 6030985 (2000-02-01), Gentile et al.
patent: 6127343 (2000-10-01), Andersen et al.
patent: 6225331 (2001-05-01), Cupps et al.
patent: 6297233 (2001-10-01), Stein et al.
patent: 6391878 (2002-05-01), Cupps et al.
patent: 6716840 (2004-04-01), Chu et al.
patent: 0343894 (1989-11-01), None
patent: WO 96/24580 (1996-08-01), None
patent: WO 97/19911 (1997-06-01), None
patent: WO 97/41119 (1997-11-01), None
patent: WO 98/07420 (1998-02-01), None
patent: WO 99/64002 (1999-12-01), None
patent: WO 00/03973 (2000-01-01), None
patent: WO 00/17191 (2000-03-01), None
patent: WO 00/74679 (2000-12-01), None
patent: WO 01/10842 (2001-02-01), None
patent: WO 01/55106 (2001-08-01), None
patent: WO 01/55107 (2001-08-01), None
patent: WO 01/55109 (2001-08-01), None
patent: WO 01/70337 (2001-09-01), None
patent: WO 01/70708 (2001-09-01), None
patent: WO 02/062776 (2002-08-01), None
patent: WO 02/081443 (2002-10-01), None
patent: WO 03/099818 (2003-12-01), None
Runti, C.; DeNardo, M. “Fusaric Acid Derivatives and Analogs as Possible Antihypertensive Drugs”, Farmaco, Edizione Scientifica (1981), 35(4), 260-8.
Wolff, M. E., “Burger's Medicinal Chemistry and Drug Discovery 5thEdition,” pp. 975-977 (1995), M. E. Wolff (ed.); published by John Wiley & Sons (New York, NY).
Banker, G. S. et al., “Modern Pharmaceutics, 3rdEdition,” pp. 596 and 451 (1996), G. S. Banker and C. T. Rhodes (eds.); published by Marcel Dekker, Inc. (New York, NY).
West, A. R., “Solid State Chemistry and Its Applications,” pp. 358 and 365 (1988), A. R. West (ed.); published by John Wiley & Sons (New York, NY).
Goodfellow, V. S. et al., “The Melanocortin System and its Role in Obesity and Cachexia,”Current Top. Med. Chem., vol. 3, No. 8, pp. 855-883 (2003); published by Bentham Science Publishers Ltd. (San Francisco, CA).
Fisher, S. L. et al., Int. J. Obes. Relat. Metab. Discord. Suppl. 1, pp. 54-48 (Feb. 1999); published by the American Dietetic Association (Chicago, IL).
Cupps et al. (1998): STN International, CAPLUS database, Columbus (Ohio), Accession No. 1998: 388504.
Julia, M. et al., “Amidines and guanidines related to congocidine. III. Urea and trazene diamidines,”Bull. Soc. Chim. Fr., No. 1, pp. 376-382, 1968, published by Masson Editeur, Paris, France.
Boyce Rustum S.
Chu Daniel
Duhl David
Renhowe Paul A.
Chiron Corporation
Friedrichsen Bernard P.
Harbin Alisa A.
Raymond Richard
Suh Young J.
LandOfFree
Guanidinobenzamides does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Guanidinobenzamides, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Guanidinobenzamides will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-3712161