Guanidine mimics as factor Xa inhibitors

Details Guanidine mimics as factor Xa inhibitors Guanidine mimics as factor Xa inhibitors

2005-06-14

2005-06-14

Raymond, Richard L. (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C514S249000, C514S266200, C514S266230, C514S300000, C514S310000, C514S313000, C514S314000, C514S373000, C514S379000, C514S395000, C514S405000, C514S406000, C544S237000, C544S258000, C544S259000, C544S260000, C544S284000, C544S293000, C546S122000, C546S143000, C546S159000, C548S207000, C548S241000, C548S304700, C548S306100, C548S362100, C548S364100, C548S364400

Reexamination Certificate

active

06906070

ABSTRACT:
The present application describes nitrogen containing heteroaromatics and derivatives thereof of formula I:or pharmaceutically acceptable salt forms thereof, wherein rings D-E represent guanidine mimics, which are useful as inhibitors of factor Xa.

REFERENCES:
patent: 5202330 (1993-04-01), Atwal et al.
patent: 5317103 (1994-05-01), Baker et al.
patent: 5342851 (1994-08-01), Sanfilippo et al.
patent: 5463071 (1995-10-01), Himmelsbach et al.
patent: 5616601 (1997-04-01), Khanna et al.
patent: 5681838 (1997-10-01), Zoller et al.
patent: 5707998 (1998-01-01), Takase et al.
patent: 5932576 (1999-08-01), Anantanarayan et al.
patent: 5998424 (1999-12-01), Galemmo et al.
patent: 6020357 (2000-02-01), Pinto et al.
patent: 6403620 (2002-06-01), Galemmo et al.
patent: 234830 (1987-09-01), None
patent: 236902 (1987-09-01), None
patent: 513387 (1992-11-01), None
patent: 554829 (1993-08-01), None
patent: 4247081 (1992-09-01), None
patent: WO 9402477 (1994-02-01), None
patent: WO 9514683 (1995-06-01), None
patent: WO 9518111 (1995-07-01), None
patent: WO 9628427 (1996-09-01), None
patent: WO 9640143 (1996-12-01), None
patent: WO 9723212 (1997-07-01), None
patent: WO 9732583 (1997-09-01), None
Tidwell et al. “Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring. Inhibitors of arginine-specific esteroproteases”, J. Med. Chem. (1978), 21(7), 613-623.

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