Griseolic acid derivatives, and their use as enzyme inhibitors

Details Griseolic acid derivatives, and their use as enzyme inhibitors Griseolic acid derivatives, and their use as enzyme inhibitors

1984-10-25

1987-01-06

Daus, Donald G.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514266, 544264, 544265, 544276, 544277, A61K 3152, C07D47300, C07D47330, C07D47334, C07D47338, C07D47340

Patent

active

046347062

ABSTRACT:
Griseolic acid derivatives of formula (I): ##STR1## wherein A represents: ##STR2## have enzyme-inhibitory activity, especially against cAMP PDE and cGMP PDE. When formulated as compositions with appropriate carriers or diluents, they may be used for the treatment of a variety of organic disorders and show toxicities less than griseolic acid itself.

REFERENCES:
patent: 3862189 (1975-01-01), Schwender
patent: 4138562 (1979-02-01), Vince
patent: 4360522 (1982-11-01), Schaeffer
patent: 4460765 (1984-07-01), Naito et al.
patent: 4479951 (1984-10-01), Klessing et al.

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