Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives
Patent
1994-06-01
1997-12-02
Kight, John
Organic compounds -- part of the class 532-570 series
Organic compounds
Carbohydrates or derivatives
514 23, 514 25, 536 185, 536 186, C07H 1520, A61K 3170
Patent
active
056937679
ABSTRACT:
Novel glycosides, especially steroidal and non-steroidal glycosides are provided. The steroidal and non-steroidal glycosides preferably are prepared from aglycons which possess valuable properties such as pharmacological properties. The glycosides are prepared from useful aglycons and possess useful properties which are the same as those of their respective unglycosylated aglycons. The glycosides are provided in acylated and deacylated form. The acylated glycosides after hydrolysis of the acyl groups possess enhanced water solubility properties, as illustrated in the case where the aglycon is acetominophen.
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Houston Todd A.
Klemke R.-Erich
Koreeda Masato
Shull Brian K.
Tuinman Roeland J.
Harrier Inc.
Kight John
Lee Howard C.
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