Glycoside compounds and production and use thereof

Details Glycoside compounds and production and use thereof Glycoside compounds and production and use thereof

1994-05-06

1996-03-05

Robinson, Douglas W.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

514885, 514886, 536 5, 536 185, 536 186, A61K 31705, C07J 900

Patent

active

054968062

ABSTRACT:
Novel glycosides 7-ketosteryl di-O-acyl-pyranoside and 7-.beta.-hydroxycholesteryl 2,3-dideoxy-.alpha.-D-erythro-hex-2-enopyranoside. The glycosides possess valuable pharmacological properties as a medicament. In particular, the cholesterol glycoside in vivo exhibits a selective cell-destructive activity on malignant cells which activity is substantially free of side effects on normal cells. The glycosides possess useful properties, especially pharmacological properties which are the same as the respective unglycosylated aglycon.

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