Glycoside compounds and methods of synthesis

Details Glycoside compounds and methods of synthesis Glycoside compounds and methods of synthesis

1997-08-21

2000-07-25

Lee, Howard C.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

514 24, 514 25, 514 26, 514 27, 514453, 536 5, 536 187, 536120, C07H 1504, A61K 3170

Patent

active

060938056

ABSTRACT:
Novel glycosides, especially steroidal and non-steroidal glycosides are provided. The steroidal and non-steroidal glycosides preferably are prepared from aglycons which possess valuable properties such as pharmacological properties. The glycosides are prepared from useful aglycons and possess useful properties which are the same as those of their respective unglycosylated aglycons. The glycosides are provided in acylated and deacylated form. The acylated glycosides after hydrolysis of the acyl groups possess enhanced water solubility properties, as illustrated in the case where the aglycon is acetominophen.

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