Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai
Reexamination Certificate
2006-06-06
2006-06-06
Barts, Samuel (Department: 1623)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Carbohydrate doai
C514S025000, C514S406000, C514S407000, C514S866000, C514S909000, C536S004100, C548S373100, C548S376100, C548S366100
Reexamination Certificate
active
07056892
ABSTRACT:
The present invention relates to glucopyranosyloxypyrazole derivatives represented by the general formula:wherein R1represents a hydrogen atom or a lower alkyl group; one of Q1and T1represents a group represented by the general formula:while the other represents a lower alkyl group or a halo(lower alkyl) group; and R2represents a hydrogen atom, a lower alkyl group, a lower alkoxy group, a lower alkylthio group, a halo(lower alkyl) group or a halogen atom, or pharmaceutically acceptable salts thereof, which have an inhibitory activity in human SGLT2 and are useful as agents for the prevention or treatment of diabetes, diabetic complications or obesity, and to pharmaceutical compositions comprising the same and intermediates thereof.
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Fujikura Hideki
Fujioka Minoru
Hiratochi Masahiro
Isaji Masayuki
Iyobe Akira
Barts Samuel
Henry Michael C.
Kissei Pharmaceutical Co. Ltd.
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