Glucopyranosyloxybenzylbenzene derivatives, medicinal...

Details Glucopyranosyloxybenzylbenzene derivatives, medicinal... Glucopyranosyloxybenzylbenzene derivatives, medicinal...

2006-05-30

2006-05-30

Wilson, James O. (Department: 1623)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

C514S035000, C536S004100, C536S018100

Reexamination Certificate

active

07053060

ABSTRACT:
The present invention relates to glucopyranosyloxybenzylbenzene derivatives represented by the general formula:wherein R1represents a hydrogen atom, a hydroxy group, a substituted or unsubstituted amino group, a carbamoyl group, a substituted or unsubstituted (lower alkyl) group, a substituted or unsubstituted (lower alkoxy) group etc.; R2represents a hydrogen atom or a lower alkyl group; and R3represents a substituted or unsubstituted (lower alkyl) group, a substituted or unsubstituted (lower alkoxy) group, a substituted or unsubstituted (lower alkylthio) group etc., or pharmaceutically acceptable salts thereof, which have an inhibitory activity in human SGLT2 and are useful as agents for the prevention or treatment of a disease associated with hyperglycemia such as diabetes, diabetic complication or obesity, pharmaceutical compositions comprising the same and intermediates thereof.

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