Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Nitrogen containing other than solely as a nitrogen in an...
Patent
1990-07-03
1992-06-30
Hollrah, Glennon H.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Nitrogen containing other than solely as a nitrogen in an...
5142385, 514331, 514427, 544162, 544163, 544165, 544170, 544177, 546194, 546246, 548561, 558303, 558391, 558419, 558422, 558426, 558430, 558431, 558432, 564230, 564237, A61K 31155, C07C27916, C07C27908, C07C29500
Patent
active
051263742
ABSTRACT:
Guanidines I ##STR1## (A=C.sub.5 -C.sub.12 -cycloalkyl which may bear up to three further substituents; benzyl substituted in the para-position; R.sup.1, R.sup.2, R.sup.3 =H, C.sub.1 -C.sub.4 -alkyl; R.sup.4 -C.sub.5 -C.sub.18 -alkyl which may be interrupted by oxygen, C.sub.5 -C.sub.18 -alkenyl, C.sub.4 -C.sub.18 -alkynyl or phenyl-C.sub.1 -C.sub.6 -alkyl, and these groups may bear up to three further substituents and the phenyl moiety of the phenylalkyl may additionally bear a phenoxy group or up to three C.sub.2 -C.sub.4 -alkenyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.6 -alkyl or haloalkyl groups, C.sub.5 -C.sub.6 -cycloalkyl-C.sub.1 -C.sub.8 -alkyl, where the ring may bear up to three further substituents; A=benzyl and R.sup.4 =C.sub.3 -C.sub.4 -alkyl which may be interrupted by oxygen, or C.sub.4 -alkenyl, both of which may bear up to three further substituents; R.sup.3 +R.sup.4 =C.sub.5 -C.sub.6 -heterocycle which may bear up to three further substituents and may be interrupted by oxygen) and the salts I.HX and the metal complexes of I.
The compounds I are suitable as fungicides.
REFERENCES:
patent: 3109859 (1963-11-01), McKay et al.
patent: 3320229 (1967-05-01), Szabo et al.
patent: 3961056 (1976-06-01), Du Charme
patent: 4427685 (1984-01-01), Stemp
Chemie der Pflanzenschutz-und Schadlingsbedampfungsmittel, 4 145-148 (1977).
J. Org. Chem. 51, 1882-1884 (1986).
J. Medicinal Chem., 12, 712-715 (1963).
Ammermann Eberhard
Lorenz Gisela
Roehl Franz
Sauter Hubert
Zipplies Matthias
BASF - Aktiengesellschaft
Hollrah Glennon H.
O'Sullivan P.
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