Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1994-12-02
1995-11-21
Robinson, Allen J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
424632, 424637, 424638, 424713, 514 35, 514 27, 514 37, 514 49, 514 80, 514114, 514140, 514146, 514147, 5142312, 514245, 514247, 514250, 514255, 514256, 514269, A61K 31535, A01N 4354, A01N 5902, A01N 5920
Patent
active
054687470
ABSTRACT:
Compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2,N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1, SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur hetero-atoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen atoms; A, B, D, E, G, U and V are independently hydrogen, halogen, C.sub.1-4 alkyl C.sub.1-4 alkoxy, cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of theforegoing being optionally substituted with one or more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano. The compounds are useful as fungicides.
REFERENCES:
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patent: 4709078 (1987-11-01), Schirmer et al.
patent: 4822908 (1989-04-01), Karbach et al.
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patent: 4863503 (1989-09-01), Anthony et al.
patent: 5124329 (1992-06-01), Clough et al.
Cheetham Rex
Clough John M.
Godfrey Christopher R. A.
Streeting Ian T.
Robinson Allen J.
Zeneca Limited
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