Fluorination process

Details Fluorination process Fluorination process

2005-12-02

2009-08-11

Price, Elvis O (Department: 1621)

Organic compounds -- part of the class 532-570 series

Organic compounds

Silicon containing

C556S476000

Reexamination Certificate

active

07572928

ABSTRACT:
Compounds of formula (II), (IIIa) or (IIIb)(variables are described in the specification) are prepared by fluorination of β,γ-unsaturated alkyl silanes. These compounds are useful as building blocks in the pharmaceutical industry.

REFERENCES:
Differding, E.; Lang, R.W.,Tetrahedron Lett. 1988, 29, 6087-6090.
Ma, J.-A.; Cahard, D.,Chem. Rev. 2004, 104, 6119-6146.
Kollonitsch, J.; Marburg, S.; Perkins, L. M.,J. Org. Chem. 1979 44, 771-777.
Gouverneur, V.; Greedy, B.Chem. Eur. J. 2002, 8, 766-771.
D. Cahard et al,Org. Lett. 2000, 2, 3699-3701.
D. Cahard et al,Tetrahedron lett. 2001, 42, 1867-1869.
Abstract of a talk given by N. Shibata Sep. 5, 2005.
Thibaudeau, S.; Fuller, R.; Gouverneur, V.Org. Biomol. Chem., 2004, 2, 1110-1112.
Hoye, T. R.; Promo, M. A.Tetrahedron Lett., 1999, 40, 1429-1432.
Burfeindt et al,J. Am. Chem. Soc., 1998, 3629-3634.
Schaffrath et al,Angew. Chem. Int. Ed., 2002, 41, 3913.
Dong et al,Nature2004, 427, 561-565.
DeYoung, J. et al,J. Chem. Soc. Chem. Commun. 1992, 811.
V. Grakauskas, A. Guest,J. Org. Chem. 1978, 43, 3485.
M. Schlosser, G. Heinz,Chem. Ber. 1969, 102, 1944.
M.J. Adam, J.M. Berry, L.D. Hall, B. D. Pate, T.J. Ruth,Can J. Chem. 61, 1983 658-660.
A. P. Lothian, C. A. Ramsden,Synlett1993, 753-755.
Takeuchi, Y. et al,J.Org. Chem., 1999, 64, 5708-5711.
B. Greedy, JM Paris, T. Vidal, V. Gouverneur,Angewandte Chemie Int. Ed. 2003, 42, 3291-3294.
Chatani et al,J. Org. Chem. 1995, 60, 1834-1840.
B. Greedy, V. Gouverneur,Chem. Commun. 2001 233-234.
G. Mentink, J. H. van Maarseveen, H. Hiemstra,Org. Lett. 2002, 4, 3497.
Nishiyama, T. et al,Tetrahedron Lett. 1998, 43-46.
W. J. Middelton,J. Org. Chem. 1975, 40, 574-578.
Gree et al,J. Org. Chem. 1996, 61, 1918.
S. Thibaudeau, V. Gouverneur,Org. Lett. 2003, 4891-4893.
Davis, F.A. et al,Tetrahedron Lett., vol. 32, No. 13, 1991, 1631-1634.
Van Overmeire, I. et al,J. Med. Chem. 1999, 42, 2697.
Van Overmeire, I. et al,J. Med. Chem. 2000, 43, 4189.
Usse et al,Tetrahedron: Asymmetry2001, 1689.
A. G. Myers, J.K. Barbay, B. Zhong,J. Am. Chem. Soc. 2001, 123, 7207.
Chamberlin et al,J. Am. Chem. Soc. 1987, 109, 672-677.
Okada et al,J. Fluorine Chemistry1997, 82, 157-161.
G. H. Posner et al,Eur. J. Org. Chem. 2003, 3889.
Kabat et al,J. Org. Chem. 2001, 66, 6141.
D. A. Evans,J. Am. Chem. Soc. 1993, 115, 6460.
L. Ghosez,J. Am. Chem. Soc. 1999, 121, 2617.
Y. Landais et al,Curr. Org. Chem. 2002, 6, 1369.
Shibata, N. et al,J. Am. Chem. Soc. 2001 123, 7001-7009.
Shibata, N. et al,J. Org. Chem. 2003, 68(6), 2494-2497.
Shibata, N. et al,J. Am. Chem. Soc. 2000, 122(43), 10728-10729.
Mohar, B. et al,Angew. Chem. Int. Ed., 2001, 40(22), 4214-4216.

Affiliated with

Also associated with

Rating

Fluorination process does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Fluorination process, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Fluorination process will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-4080252