Fluorinated diazabicycloalkane derivatives

Details Fluorinated diazabicycloalkane derivatives Fluorinated diazabicycloalkane derivatives

1990-09-20

1992-02-04

Berch, Mark L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Nitrogen attached directly or indirectly to the purine ring...

540472, 540556, 568775, 568364, 568656, 570261, 570123, C07D48708, C07D51900, C07B 3900

Patent

active

050861786

ABSTRACT:
Fluorinated diazabicycloalkane derivative of the following Formula I: ##STR1## wherein n represents 0, 1 or 2; R represents a quaternizing organic group; each R.sup.1, R.sup.2, R.sup.3, R.sup.4 and R.sup.5 independently represents hydrogen, C.sub.1 -C.sub.6 alkyl, aryl, C.sub.1 -C.sub.6 alkyl-substituted aryl or aryl-substituted C.sub.1 -C.sub.6 alkyl and each X.sup.- independently represents a conterion or 2X.sup.- represents a single divalent counterion, are electrophilic fluorinating agents.

REFERENCES:
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