Epinine esters and pharmaceutical compositions thereof

Details Epinine esters and pharmaceutical compositions thereof Epinine esters and pharmaceutical compositions thereof

1977-07-28

1980-08-19

Myers, Jane S.

Drug, bio-affecting and body treating compositions

Antigen, epitope, or other immunospecific immunoeffector

Recombinant or stably-transformed bacterium encoding one or...

560142, C07C 9326, A61K 31215

Patent

active

042184703

ABSTRACT:
Novel cardiocirculatory analeptics are prepared, which are epinine esters as obtained by reacting epinine (N-methyldopamine) with branched-chain aliphatic carboxylic acids. Exemplary members are 3,4-di-O-butyrylepinine and 3,4-di-O-pivaloylepinine. These medicaments are effective also by the oral route of administration, contrary to the hitherto commonly used dopamine derivatives which are rapidly destroyed by metabolization when administered orally.

REFERENCES:
patent: 2400038 (1946-05-01), Buck
patent: 3809714 (1974-05-01), Hussain et al.
patent: 3868461 (1975-02-01), Hussain et al.
patent: 4031242 (1977-06-01), Jones et al.

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