Enhanced electrotransport of therapeutic agents having polybasic

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424400, 424448, 424449, 514788, 514772, 514318, A61K 970

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active

060045779

ABSTRACT:
Improved electrotransport of therapeutic agents which include agent cations and polybasic anionic counterions. Improved electrotransport is obtained by treating the therapeutic agent with a multivalent metal compound of the formula MX where M is a metallic cation having a valency of at least +2 and is reactive with the polybasic anionic counter ion and X is a pH-increasing anion. Reduction in species which compete with the therapeutic agent for electrotranport is obtained.

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