Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1998-10-05
1999-10-05
Richter, Johann
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
548247, 558375, 564163, 564244, 564246, C07D26102, C07D26108, C07C25718
Patent
active
059626933
ABSTRACT:
The present invention relates to processes for the conversion of nitrites to amidines in the preparation of compounds which are antagonists of the platelet glycoprotein IIb/IIIa fibrinogen receptor complex. The compounds described herein are potent thrombolytics and useful for the inhibition of platelet aggregation in the treatment of thromboembolic disorders.
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Confalone Pasquale N.
Li Hui-Yin
Ma Philip
DuPont Pharmaceuticals Company
Oswecki Jane C.
Richter Johann
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