Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai
Reexamination Certificate
2005-08-30
2009-06-23
Tate, Christopher R. (Department: 1654)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Peptide containing doai
C514S008100, C530S317000
Reexamination Certificate
active
07550428
ABSTRACT:
A complex of an echinocandin compound with a carbohydrate is described having improved thermal stability and water solubility. A process for making the echinocandin/carbohydrate complex is also described as well as the use of the complex in pharmaceutical formulations and treatments of fungal infections.
REFERENCES:
patent: 3293482 (1966-12-01), Wolkstein
patent: 3978210 (1976-08-01), Mizuno et al.
patent: 4293482 (1981-10-01), Abbott et al.
patent: 4293483 (1981-10-01), Debono
patent: 4293489 (1981-10-01), Debono
patent: 4299763 (1981-11-01), Abbott et al.
patent: 4304716 (1981-12-01), Abbott et al.
patent: 4320052 (1982-03-01), Abbott et al.
patent: 4348384 (1982-09-01), Horikoshi et al.
patent: 4876241 (1989-10-01), Feldman et al.
patent: 4927831 (1990-05-01), Malamas
patent: 5141674 (1992-08-01), Leigh
patent: 5166135 (1992-11-01), Schmatz
patent: 5198421 (1993-03-01), Chen et al.
patent: 5202309 (1993-04-01), Schwartz et al.
patent: 5376634 (1994-12-01), Iwamoto et al.
patent: 5541160 (1996-07-01), Balkovec et al.
patent: 5573936 (1996-11-01), Kreuzman et al.
patent: 5618787 (1997-04-01), Jamison et al.
patent: 5629289 (1997-05-01), Rodriguez
patent: 5629290 (1997-05-01), LaGrandeur et al.
patent: 5646111 (1997-07-01), Borromeo et al.
patent: 5652213 (1997-07-01), Jamison et al.
patent: 5693611 (1997-12-01), Henle et al.
patent: 5696084 (1997-12-01), Lartey et al.
patent: 5741775 (1998-04-01), Balkovec et al.
patent: 5786325 (1998-07-01), Borromeo et al.
patent: 5932543 (1999-08-01), Burkhardt et al.
patent: 5952008 (1999-09-01), Backstrom et al.
patent: 5965525 (1999-10-01), Burkhardt et al.
patent: 5972996 (1999-10-01), Nielsen-Kahn et al.
patent: 5985309 (1999-11-01), Edwards et al.
patent: 5993805 (1999-11-01), Sutton et al.
patent: 6001336 (1999-12-01), Gordon
patent: 6043341 (2000-03-01), Udodong et al.
patent: 6153224 (2000-11-01), Staniforth
patent: 6258821 (2001-07-01), Stogniew et al.
patent: 6267958 (2001-07-01), Andya et al.
patent: 6284277 (2001-09-01), Bouloumie et al.
patent: 6284282 (2001-09-01), Maa et al.
patent: 6309623 (2001-10-01), Weers et al.
patent: 6323176 (2001-11-01), Jamison et al.
patent: 6384013 (2002-05-01), Burkhardt et al.
patent: 6433040 (2002-08-01), Dellamary et al.
patent: 6451349 (2002-09-01), Robinson et al.
patent: 6475523 (2002-11-01), Staniforth
patent: 6506726 (2003-01-01), Dobbins et al.
patent: 6565885 (2003-05-01), Tarara et al.
patent: 6590073 (2003-07-01), Dalder et al.
patent: 6638495 (2003-10-01), Kabalnov et al.
patent: 6653281 (2003-11-01), Borromeo et al.
patent: 6660843 (2003-12-01), Feige et al.
patent: 6670324 (2003-12-01), Jamison et al.
patent: 6689390 (2004-02-01), Bernstein et al.
patent: 6709650 (2004-03-01), Sutton et al.
patent: 6743777 (2004-06-01), Burkhardt et al.
patent: 6916784 (2005-07-01), Burkhardt et al.
patent: 6960564 (2005-11-01), Milton et al.
patent: 7041637 (2006-05-01), Larew et al.
patent: 2002/0151474 (2002-10-01), Schwier et al.
patent: 2002/0161176 (2002-10-01), Dalder et al.
patent: 2003/0039667 (2003-02-01), Jira et al.
patent: 2003/0054981 (2003-03-01), Milton et al.
patent: 2003/0104048 (2003-06-01), Patel et al.
patent: 2003/0220236 (2003-11-01), Burkhardt et al.
patent: 2004/0223997 (2004-11-01), Stogniew
patent: 2043762 (1991-12-01), None
patent: 2803581 (1979-08-01), None
patent: 0031221 (1981-07-01), None
patent: 0032009 (1981-07-01), None
patent: 0359529 (1990-03-01), None
patent: 0359529 (1990-03-01), None
patent: 0365324 (1990-04-01), None
patent: 0365324 (1990-04-01), None
patent: 0447186 (1991-09-01), None
patent: 0448343 (1991-09-01), None
patent: 0448343 (1991-09-01), None
patent: 0448353 (1991-09-01), None
patent: 0448353 (1991-09-01), None
patent: 0448354 (1991-09-01), None
patent: 0448354 (1991-09-01), None
patent: 0448355 (1991-09-01), None
patent: 0448355 (1991-09-01), None
patent: 0448356 (1991-09-01), None
patent: 0448356 (1991-09-01), None
patent: 0460882 (1991-12-01), None
patent: 0460882 (1991-12-01), None
patent: 0460882 (1991-12-01), None
patent: 0462531 (1991-12-01), None
patent: 0462531 (1991-12-01), None
patent: 0486011 (1992-05-01), None
patent: 0486011 (1992-05-01), None
patent: 0503960 (1992-09-01), None
patent: 0525889 (1993-02-01), None
patent: 0561639 (1993-09-01), None
patent: 0561639 (1993-09-01), None
patent: 0589074 (1994-03-01), None
patent: 0744405 (1996-11-01), None
patent: 0757058 (1997-02-01), None
patent: 0931834 (1999-07-01), None
patent: 2241956 (1991-09-01), None
patent: 2242194 (1991-09-01), None
patent: 03240727 (1991-10-01), None
patent: 05271097 (1993-10-01), None
patent: 5271097 (1993-10-01), None
patent: 06172205 (1994-06-01), None
patent: 61772205 (1994-06-01), None
patent: WO 9637512 (1991-11-01), None
patent: WO 9425048 (1994-11-01), None
patent: WO 9527074 (1995-10-01), None
patent: WO 9631228 (1996-10-01), None
patent: WO 9637509 (1996-11-01), None
patent: WO 9637510 (1996-11-01), None
patent: WO 9637511 (1996-11-01), None
patent: WO 9705163 (1997-02-01), None
patent: WO 9727864 (1997-08-01), None
patent: WO 9730695 (1997-08-01), None
patent: WO 9906062 (1999-02-01), None
patent: WO 9943337 (1999-09-01), None
patent: WO 0011023 (2000-03-01), None
patent: WO 0011023 (2000-03-01), None
patent: WO 0012540 (2000-03-01), None
patent: WO 0034315 (2000-06-01), None
patent: WO 0034315 (2000-06-01), None
patent: WO 0035944 (2000-06-01), None
patent: WO 0035945 (2000-06-01), None
patent: WO 0051564 (2000-09-01), None
patent: WO 0051567 (2000-09-01), None
patent: WO 0052036 (2000-09-01), None
patent: WO 0052037 (2000-09-01), None
patent: WO 03105767 (2003-12-01), None
Avis, K. E. (1990). “Parenteral Preparations” Chapter 84In Remington Pharmaceutical Sciences. 18thedition, Mack Publishing Company pp. 1545-1569.
Longer, M. A. and Robinson, J. R. (1990). “Transdermal Systems” in Chapter 91In Remington Pharmaceutical Sciences, 18thedition, Mack Publishing Company. pp. 1690-1693.
Nema, S. et al. (1997). “Excipients and Their Use in Injectable Products,”PDA Journal of Pharm. Science and Tech. 51(4):166-171.
Sclarra, J. J. and Cutie, A. J. (1990), “Aerosols” Chapter 92In Remington Pharmaceutical Sciences. 18thedition, Mack Publishing Company. pp. 1694-1712.
Turco, S. J. (1990). “Intravenous Admixtures,” Chapter 85In Remington Pharmaceutical Sciences. 18thedition, Mack Publishing Company. pp. 1570-1580.
Ibrahim, F. S. et al., (1995) “The effort of pH, sugars and calcium ion concentration on the thermal stability of whey proteins”Egyptian J. Dairy Sci. 23:177-178.
Nail, S. L. and Fatlin, L. A. (1993) “Chapter 3: Freeze drying: Principles and practice”Pharmaceutical Dosage Forms, Parenteral Medications, vol. 2, 2ndEdition, edited by Kenneth, E. A. et al., Marcel Dekker, Inc., pp. 163-233.
Etter, M. C. and Baures, P.W. (1988) “Triphenyloposphine Oxide as a Crystallization Aid,”J. Am. Chem. Soc. 110:639-640.
Debono, M. et al. Al, (1995), “Semisynthetic Chemical Modification of the Antifungal Lipopeptide Echinocandin B (ECB): Structure-Activity Studies of the Lipophilic and Geometric Parameters of Polyarylated Acyl Analogs of ECB,”J Med Chem. 38(17):3271-3281.
Groll, A.H. et al. (2001), “Pharmacokinetic and Pharmacodynamic Modeling of Anidulafungin (LY303366): Reappraisal of its Efficacy in neutropenic Animal Models of Opportunistic Mycoses Using Optical Plasma Sampling,”Antimicrobial Agents and Chemotherapy45(10):2845-2855. International Search Report mailed on Dec. 9, 2003, for PCT Patent Application No. PCT/US03/18754 filed on Jun. 12, 2003, 5 pages.
International Search Report for PCT Application No. PCT/US00/05494 filed Mar. 2, 2000, mailed Jun. 7, 2000, three pages.
International Search Report for PCT Application No. PCT/US00/05508 filed Mar. 2, 2000, mailed Aug. 21, 2000, two pages.
International Search Report for PCT Application No. PCT/US00/05546 filed Mar. 2, 2000, mailed Aug. 11, 2000, three pages.
International Search Report for PCT Application No. PCT/US00/05547 filed Mar. 2, 2000, mailed Jul. 19, 2000
Larew Larry A.
Milton Nathaniel
Moder Kenneth Philip
Sabatowski James Lawrence
Eli Lilly and Company
Tate Christopher R.
Tebbutt Jason G.
Teller Roy
Zelson Steve T.
LandOfFree
Echinocandin/carbohydrate complexes does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Echinocandin/carbohydrate complexes, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Echinocandin/carbohydrate complexes will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-4117862