Eburnamonine oxime derivatives, salts thereof, and pharmaceutica

Details Eburnamonine oxime derivatives, salts thereof, and pharmaceutica Eburnamonine oxime derivatives, salts thereof, and pharmaceutica

1985-06-03

1988-04-05

Daus, Donald G.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514283, 514237, 544361, 544125, 546 51, A61K 3144, C07D46100

Patent

active

047359439

ABSTRACT:
There is disclosed novel eburnamonine oxime, its derivatives and salts, process for the manufacture thereof and pharmaceutical agents containing the same. The compounds are represented by the following formula. ##STR1## wherein R is hydrogen, alkyl, alkoxyalkyl, or oxisilanylalkyl group or a group of ##STR2## R.sup.1 and R.sup.2 are same or different and respectively hydrogen, alkyl having 1 to 4 carbon atoms, aryl or aralkyl group, or R.sup.1 represents together with R.sup.2 and the neighboring nitrogen atom a non-substituted or substituted heterocyclic ring, and n is an integer of 2 or 3.

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