Disaccharide sialidase substrates and inhibitors

Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives

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536 171, 536 175, 536 53, 536 54, 536 55, 536 551, 536116, 536118, 536119, 536120, 536121, 536122, 5361231, 53612313, C07H 504, C07H 510

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active

054896754

ABSTRACT:
Novel NeuAc-Gal dissacharide sialidase substrates and inhibitors which are locked into rigid conformation by the attachment of an alkyl group at the C-6 arm of the galactose core are provided. Also provided is a method for the inhibition of sialidase activity.

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