Dipeptidyl peptidase-IV inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S235500, C514S381000, C514S408000, C544S111000, C544S132000, C544S152000, C548S250000, C548S530000

Reexamination Certificate

active

08076330

ABSTRACT:
The present invention relates generally to pyrrolidine and thiazolidine DPP-IV inhibitor compounds. The present invention also provides synthetic methods for preparation of such compounds, methods of inhibiting DPP-IV using such compounds and pharmaceutical formulations containing them for treatment of DPP-IV mediated diseases, in particular, Type-2 diabetes.

REFERENCES:
patent: 3297709 (1967-01-01), Davis et al.
patent: 5064853 (1991-11-01), Gasc et al.
patent: 5118811 (1992-06-01), Uchida et al.
patent: 5254543 (1993-10-01), Hanko et al.
patent: 5262386 (1993-11-01), Lüthy et al.
patent: 5338860 (1994-08-01), Baasner et al.
patent: 5391556 (1995-02-01), Heckel et al.
patent: 5407950 (1995-04-01), Okubo et al.
patent: 5437969 (1995-08-01), Schmuck et al.
patent: 5445928 (1995-08-01), Schmuck et al.
patent: 5475016 (1995-12-01), Hanko et al.
patent: 5482920 (1996-01-01), Lüthy
patent: 5492916 (1996-02-01), Morriello et al.
patent: 5492920 (1996-02-01), Chen et al.
patent: 5494919 (1996-02-01), Morriello et al.
patent: 5514505 (1996-05-01), Limburg et al.
patent: 5563014 (1996-10-01), Malhotra et al.
patent: 5569662 (1996-10-01), Satake et al.
patent: 5618808 (1997-04-01), Nagel
patent: 5622973 (1997-04-01), Morriello et al.
patent: 5627285 (1997-05-01), Hanko et al.
patent: 5665719 (1997-09-01), Bock et al.
patent: 5674905 (1997-10-01), Kalindjian et al.
patent: 5714471 (1998-02-01), Rowe et al.
patent: 5767097 (1998-06-01), Tam
patent: 5795894 (1998-08-01), Shue et al.
patent: 5804560 (1998-09-01), McDonald et al.
patent: 5914150 (1999-06-01), Porter et al.
patent: 5939560 (1999-08-01), Jenkins et al.
patent: 5962419 (1999-10-01), McDonald et al.
patent: 5968929 (1999-10-01), Blythin et al.
patent: 5969100 (1999-10-01), Munoz et al.
patent: 6011155 (2000-01-01), Villhauer
patent: 6015879 (2000-01-01), McDonald et al.
patent: 6017929 (2000-01-01), Tanaka et al.
patent: 6051575 (2000-04-01), Blythin et al.
patent: 6051684 (2000-04-01), McDonald et al.
patent: 6057314 (2000-05-01), Dimaio et al.
patent: 6110909 (2000-08-01), Yukimasa et al.
patent: 6124305 (2000-09-01), Villhauer
patent: 6153171 (2000-11-01), Rowe et al.
patent: 6166063 (2000-12-01), Villhauer
patent: 6180698 (2001-01-01), Porter et al.
patent: 6191161 (2001-02-01), Kánai et al.
patent: 6201132 (2001-03-01), Jenkins et al.
patent: 6207668 (2001-03-01), Braun et al.
patent: 6228885 (2001-05-01), Palla et al.
patent: 6303661 (2001-10-01), Demuth et al.
patent: 6316486 (2001-11-01), Lieb et al.
patent: 6319902 (2001-11-01), Sugawara et al.
patent: 6331537 (2001-12-01), Hamilton et al.
patent: 6337340 (2002-01-01), Ross et al.
patent: 6358887 (2002-03-01), Fischer et al.
patent: 6358991 (2002-03-01), Jenkins
patent: 6369051 (2002-04-01), Jenkins
patent: 6376486 (2002-04-01), Jenkins et al.
patent: 6380246 (2002-04-01), Lieb et al.
patent: 6380398 (2002-04-01), Kanstrup et al.
patent: 6387893 (2002-05-01), Evans
patent: 6432969 (2002-08-01), Villhauer
patent: 6455502 (2002-09-01), Bryant et al.
patent: 6455568 (2002-09-01), Jenkins et al.
patent: 6465454 (2002-10-01), Jenkins et al.
patent: 6476026 (2002-11-01), Bryant et al.
patent: 6500885 (2002-12-01), Porter et al.
patent: 6509332 (2003-01-01), Jenkins
patent: 6518299 (2003-02-01), Chand et al.
patent: 6521644 (2003-02-01), Broqua
patent: 6537987 (2003-03-01), Hamanaka et al.
patent: 6559163 (2003-05-01), Cai et al.
patent: 6583170 (2003-06-01), Pickar et al.
patent: 6593327 (2003-07-01), Bryant et al.
patent: 6613761 (2003-09-01), Yukimasa et al.
patent: 6635658 (2003-10-01), Madera et al.
patent: 6635660 (2003-10-01), Jenkins et al.
patent: 6645995 (2003-11-01), Kanstrup et al.
patent: 6673815 (2004-01-01), Devasthale et al.
patent: 6706742 (2004-03-01), De Nanteuil et al.
patent: 6713487 (2004-03-01), Yu et al.
patent: 6716843 (2004-04-01), De Nanteuil et al.
patent: 6746990 (2004-06-01), Fischer et al.
patent: 6767864 (2004-07-01), Fischer et al.
patent: 6774112 (2004-08-01), Gougoutas
patent: 6777414 (2004-08-01), Shiotani et al.
patent: 6803357 (2004-10-01), Bachovchin et al.
patent: 6806278 (2004-10-01), Madera et al.
patent: 6861440 (2005-03-01), Boehringer et al.
patent: 6911467 (2005-06-01), Evans
patent: 2001/0025023 (2001-09-01), Carr
patent: 2001/0031780 (2001-10-01), Kanstrup et al.
patent: 2002/0006899 (2002-01-01), Pospisilik et al.
patent: 2002/0016318 (2002-02-01), Miller
patent: 2002/0019373 (2002-02-01), Jenkins et al.
patent: 2002/0019377 (2002-02-01), Jenkins et al.
patent: 2002/0019391 (2002-02-01), Jenkins et al.
patent: 2002/0019392 (2002-02-01), Jenkins
patent: 2002/0019433 (2002-02-01), Jenkins
patent: 2002/0022617 (2002-02-01), Adelman et al.
patent: 2002/0022618 (2002-02-01), Jenkins et al.
patent: 2002/0022619 (2002-02-01), Bakthavatachalam
patent: 2002/0025952 (2002-02-01), Jenkins et al.
patent: 2002/0028792 (2002-03-01), Jenkins et al.
patent: 2002/0028800 (2002-03-01), Jenkins et al.
patent: 2002/0042432 (2002-04-01), Jenkins
patent: 2002/0045641 (2002-04-01), Hamilton et al.
patent: 2002/0052510 (2002-05-01), Hamilton et al.
patent: 2002/0052514 (2002-05-01), Hamilton et al.
patent: 2002/0086996 (2002-07-01), Bryant et al.
patent: 2002/0103384 (2002-08-01), Kanstrup et al.
patent: 2002/0128305 (2002-09-01), Jenkins et al.
patent: 2002/0161008 (2002-10-01), Cai et al.
patent: 2002/0165164 (2002-11-01), Demuth et al.
patent: 2002/0193390 (2002-12-01), Villhauer
patent: 2002/0198205 (2002-12-01), Himmelsbach et al.
patent: 2002/0198242 (2002-12-01), Demuth et al.
patent: 2003/0008905 (2003-01-01), Demuth et al.
patent: 2003/0032625 (2003-02-01), Jensen et al.
patent: 2003/0045432 (2003-03-01), Fischer et al.
patent: 2003/0064935 (2003-04-01), Gougoutas
patent: 2003/0069169 (2003-04-01), Macor et al.
patent: 2003/0073701 (2003-04-01), Thompson et al.
patent: 2003/0078247 (2003-04-01), De Nanteuil et al.
patent: 2003/0087950 (2003-05-01), DeNanteuil et al.
patent: 2003/0092732 (2003-05-01), Yu et al.
patent: 2003/0096796 (2003-05-01), Bryant et al.
patent: 2003/0096827 (2003-05-01), Yu et al.
patent: 2003/0096857 (2003-05-01), Evans
patent: 2003/0114389 (2003-06-01), Webb
patent: 2003/0119750 (2003-06-01), Demuth et al.
patent: 2003/0119788 (2003-06-01), Bryant et al.
patent: 2003/0125304 (2003-07-01), Demuth et al.
patent: 2003/0130199 (2003-07-01), von Hoersten et al.
patent: 2003/0130281 (2003-07-01), Boehringer et al.
patent: 2003/0130306 (2003-07-01), Devasthale et al.
patent: 2003/0135023 (2003-07-01), Demuth et al.
patent: 2003/0139434 (2003-07-01), Balkan et al.
patent: 2003/0148961 (2003-08-01), Heiser et al.
patent: 2003/0153509 (2003-08-01), Bachovchin et al.
patent: 2003/0162820 (2003-08-01), Demuth et al.
patent: 2003/0166578 (2003-09-01), Arch et al.
patent: 2003/0171362 (2003-09-01), Madera et al.
patent: 2003/0175350 (2003-09-01), Sugita et al.
patent: 2003/0176357 (2003-09-01), Pospisilik et al.
patent: 2003/0199527 (2003-10-01), Hamanaka et al.
patent: 2003/0203890 (2003-10-01), Steiner et al.
patent: 2003/0216450 (2003-11-01), Evans et al.
patent: 2003/0225102 (2003-12-01), Sankaranarayanan
patent: 2003/0232985 (2003-12-01), Thompson et al.
patent: 2004/0002495 (2004-01-01), Sher et al.
patent: 2004/0002519 (2004-01-01), Damon et al.
patent: 2004/0009877 (2004-01-01), Fischer et al.
patent: 2004/0048867 (2004-03-01), Cai et al.
patent: 2004/0058876 (2004-03-01), Hoffmann et al.
patent: 2004/0063935 (2004-04-01), Yasuda et al.
patent: 2004/0072819 (2004-04-01), Yukimasa et al.
patent: 2004/0072892 (2004-04-01), Fukushima et al.
patent: 2004/0077601 (2004-04-01), Adams et al.
patent: 2004/0077645 (2004-04-01), Himmelsbach et al.
patent: 2004/0077761 (2004-04-01), Pavez Aranguiz
patent: 2004/0082497 (2004-04-01), Evans et al.
patent: 2004/0082607 (2004-04-01), Oi et al.
patent: 2004/0082622 (2004-04-01), Hamilton et al.
patent: 2004/0087587 (2004-05-01), Himmelsbach et al.
patent: 2004/0092604 (2004-05-01), Madera et al.
patent: 2004/0106655 (2004-06-01), Kitajima et al.
patent: 2004/0106802 (2004-06-01), Sankaranarayanan
patent: 2004/0121964 (2004-06-01), Madar et al.
patent: 2004/0121994 (2004-06-01)

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