Drug – bio-affecting and body treating compositions – Antigen – epitope – or other immunospecific immunoeffector – Bacterium or component thereof or substance produced by said...
Patent
1982-02-18
1982-12-07
Bond, Robert T.
Drug, bio-affecting and body treating compositions
Antigen, epitope, or other immunospecific immunoeffector
Bacterium or component thereof or substance produced by said...
2602393T, 2602393B, A61K 3155, C07D47114
Patent
active
043627323
ABSTRACT:
There is presented imidazodiazepines of the formula ##STR1## wherein A together with the two carbon atoms denoted as .alpha. and .beta. is a pyridine ring, X is an oxygen or sulphur atom, R.sup.1 is hydrogen, halogen, lower alkyl, lower alkoxymethyl or the group--COOR.sup.3 and R.sup.2 and R.sup.3 each are lower alkyl, and their pharmaceutically acceptable acid addition salts. The compounds are useful in the antagonization of the central-depressant, muscle relaxant, ataxic, blood pressure-lowering and respiratory-depressant properties of 1,4-benzodiazepines which have tranquillizing activity, for example as antidotes in the case of intoxications with 1,4-benzodiazepines which have tranquillizing activity.
Also presented are methods to produce such imidazodiazepines.
REFERENCES:
patent: 4316832 (1982-02-01), Gerecke et al.
Hunkeler Walter
Kyburz Emilio
Bond Robert T.
Hoffman Frank P.
Hoffmann-La Roche Inc.
Leon Bernard S.
Saxe Jon S.
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