Derivatives of substituted imidazo benzoxazin-1-one and process

Details Derivatives of substituted imidazo benzoxazin-1-one and process Derivatives of substituted imidazo benzoxazin-1-one and process

1993-06-03

1994-11-15

Richter, Johann

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514872, 544102, C07D48704, A61K 3500

Patent

active

053648544

ABSTRACT:
Derivatives of 2,3,3a,4-tetrahydro-2-azabicyclo alkyl-1H-imidazo[5,1,-c][1,4]benzoxazin-1-one are provided of general formula (I) ##STR1## in which inter alia R.sub.3 represents ##STR2## wherein n is an integer of 1 or 2 and R.sub.8 is hydrogen, C.sub.1 -C.sub.6 alkyl unsubstituted or substituted by phenyl, C.sub.2 -C.sub.4 alkenyl, C.sub.2 -C.sub.4 alkynyl, formyl or C.sub.2 -C.sub.6 alkanoyl; and the pharmaceutically acceptable salts thereof, which are useful in the treatment of CNS disorders, gut motility disorders, emesis and migraine, as cognition activators, anti-drug addiction agents and analgesic.

REFERENCES:
Heterocycles 1986, 24 (12), 3483-8; C.A.: 107:58949k.
WO-9107408-Novo Nordisk A/S-priority Nov. 22, 1989, published on May 30, 1991-Derwent 91-178035.

Affiliated with

Also associated with

Rating

Derivatives of substituted imidazo benzoxazin-1-one and process does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Derivatives of substituted imidazo benzoxazin-1-one and process , we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Derivatives of substituted imidazo benzoxazin-1-one and process will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-1097903