Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2009-07-17
2011-10-25
Shameem, Golam M (Department: 1622)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C546S112000, C546S113000, C514S299000
Reexamination Certificate
active
08044066
ABSTRACT:
The invention relates to compounds of formula (I):Wherein n, the pyrrolopyridine core, X, Y and W are as described herein. The invention also relates to a preparation method and to a therapeutic application.
REFERENCES:
patent: 7745467 (2010-06-01), Dubois et al.
patent: 7763636 (2010-07-01), Dubois et al.
patent: WO 03/049702 (2003-06-01), None
patent: WO 03/068749 (2003-08-01), None
patent: WO 2004/104001 (2004-12-01), None
patent: WO 2005/080391 (2005-09-01), None
patent: WO 2006/059163 (2006-06-01), None
patent: WO 2006/089309 (2006-08-01), None
patent: WO 2007/088277 (2007-08-01), None
Abramovitch, R. A., et. al., Microwave-Assisted Alkylations of Activatived Methylene Groups, Synthetic Communications, (1995), vol. 25, No. 1, pp. 1-8.
Antilla, J. C. et al, The Copper-Catalyzed N-Arylation of Indoles, J. Am. Chem. 'Soc., vol. 124, No. 30, (2002), pp. 11684-11688.
Barberis. C., et. al., Cu(I)-Catalyzed intramolecular Cyclization of Ene-Carbamates: Synthesis of indoles and Pyrrole[2,3-c]Pyridines, Tetrahedron Letters, vol. 46, (2005), pp. 8877-8880.
Fagan, G. P., et. al., Indoline Analogues of Idazoxan: Potent a2-Antagonists and a1-Agonists, J. Med. Chem., (1988), vol. 31, pp. 944-948.
Fresneda, P. M., et. al., Synthetic Studies Towards the 2-Aminopyrimidine Alkaloids Variolins and Meridianins From Marine Chain, Tetrahedron Letters, vol. 41, (2000), pp. 4777-4780.
Frydman, B., et. al., Pyrroles From Azaindoles. A Synthesis of Porphobilinogen, J. Am. Chem. Soc., (1965), vol. 87, pp. 3530-3531.
Frydman. B., et. al., Synthesis of Substituted 4- and 6-Azaindoles, J.Org.Cnem., vol. 33, No. 10, (1968), pp. 3762-3766.
Furstner A., et. al., Ion-Catalyzed Cross-Coupling Reactions, J. Am Chem Soc., (2002), vol. 124. pp. 13856-13863.
Klapars, A., et. al., A General and Efficient Copper Catalyst for the Amidation of Aryl Halides and the N-Arylation of Nitrogen Heterocycles, J. Am. Chem, Soc., (2001) pp, 7727-7729 vol. 123.
Kolasa, T, et. al., Synthesis of Indolylalkoxyiminoalkylcarboxylates as Leukotriene Biosynthesis Inhibitors, Bioorganic & Medicinal Chemistry, vol. 5, No. 3, pp. 507-514, (1997).
Lachance, N., et. al., Rapid and Efficient Microwave-Assisted Synthesis of 4-, 5-. 6-, and 7-Azaindoles, Synthesis, (2005), vol. 15, pp. 2571-2577.
Lomberget, T., et. al., A Regioselective Route to 5- and 6-Azaindoles, Synlett, (2005), vol. 13, pp. 2080-2082.
Mitsunobu, O., et. al., The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products, Synthesis, (1981), pp. 1-28.
Nazare, M., et. al., A Flexible, Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Chloroanilines and Chloroaminopyridines With Ketones, Angew. Chem. Int. Ed., (2004), vol. 43, pp. 4526-4528.
Roy, P. J., et. al., The Hemetsberger-Knittel Synthesis of Substituted 5-, 6-, and 7-Azaindotes, Synthesis, (2005), vol, 16. pp. 2751-2757.
Trecourt, F., et al., First Syntheses of Caerulomycin E and Collismycins A and C. A New Synthesis of Caerulomycin A, J. Org. Chem., (1998). vol. 63, pp. 2892-2897.
Yakhontov, L. N., et. al., About Reactivity of Isomeric Azaindoles, Tetrahedron Letters, No. 24, pp. 1909-1912, (1969).
Dubois Laurent
Evanno Yannick
Malanda André
Sanofi-Aventis
Scully , Scott, Murphy & Presser, P.C.
Shameem Golam M
LandOfFree
Derivatives of pyrrolopyridine-2-carboxamides, preparation... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Derivatives of pyrrolopyridine-2-carboxamides, preparation..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Derivatives of pyrrolopyridine-2-carboxamides, preparation... will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-4267284