Derivative-compound-conjugates and pharmaceutical compositions c

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai

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514178, 514182, 536 5, 540106, A61K 3170, A61K 3156, C07J 1700, C07J 4100

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active

055717950

ABSTRACT:
Novel glycosylated steroid derivatives for facilitating the transport of compounds across biological membranes, either in admixture or as conjugates, are disclosed. A novel process for efficient synthesis of these glycosylated steroid derivatives, using activated glycosyl sulfoxide intermediates is also provided.

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