Organic compounds -- part of the class 532-570 series – Organic compounds – Carbohydrates or derivatives
Patent
1980-06-12
1982-03-23
Brown, Johnnie R.
Organic compounds -- part of the class 532-570 series
Organic compounds
Carbohydrates or derivatives
424180, 435 76, A61K 3171, C07H 1708
Patent
active
043213626
ABSTRACT:
23-De(mycinosyloxy)tylosin (DMOT) which has the formula: ##STR1## 20-dihydro-DMOT, specified acyl ester derivatives, and the acid addition salts thereof are useful antibacterial agents. New methods of making 23-deoxy-5-O-my-caminosyltylonolide (DOMT) and 20-dihydro-DOMT by mild acid hydrolysis of DMOT and 20-dihydro-DMOT, respectively, are included.
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Baltz Richard H.
Seno Eugene T.
Wild Gene M.
Brown Johnnie R.
Eli Lilly and Company
Harrison Nancy J.
Whale Arthur R.
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