Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1998-10-27
2000-08-15
Richter, Johann
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
548182, 548200, 548213, 548214, 548524, 548527, C07D20712, C07D20724, C07D40312
Patent
active
061039101
ABSTRACT:
New compounds have the formula: ##STR1## wherein R, R.sup.1, X and Y have the meanings described herein. Methods are set forth for synthesizing these compounds and using these compounds to treat diseases associated with amyloidosis, such as Alzheimer's disease, maturity onset diabetes mellitus, familial amyloid polyneuropathy, scrapie, and Kreuzfeld-Jacob disease.
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Hertel Cornelia
Hoffmann Torsten
Jakob-Roetne Roland
Norcross Roger David
Epstein William H.
Hoffmann-La Roche Inc.
Johnston George W.
Oswecki Jane C.
Parise John P.
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