Cyclosporine derivatives and uses thereof

Chemistry: natural resins or derivatives; peptides or proteins; – Peptides of 3 to 100 amino acid residues – Cyclic peptides

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514 9, 514 11, 514 15, 530327, 4241931, A61K 3812, A61K 3800, C07D 1600, C07D 1700

Patent

active

059902744

ABSTRACT:
The present invention provides novel cyclosporine C (CsC) derivatives having improved protein conjugatibility and hydrolytic stability. The present invention further provides a CsC derivative conjugated to a carrier, e.g., a solid support. Preferably, the solid support is a latex or magnetic particle.

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