Cyclopentane(ene) heptenoic or heptanoic acids and derivatives t

Details Cyclopentane(ene) heptenoic or heptanoic acids and derivatives t Cyclopentane(ene) heptenoic or heptanoic acids and derivatives t

1993-12-28

1996-08-13

Raymond, Richard L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Ester doai

514573, 514613, 514659, 514729, 560121, 562503, 562504, 562510, 564189, 564453, 564454, 568838, A61K 3125, A61K 31557, C07C40500, C07C23300

Patent

active

055456650

ABSTRACT:
The invention relates to 7-[5-hydroxy-2-(hydroxyhydrocarbyl or heteroatom-substituted hydroxy hydrocarbyl)-3-hydroxycyclopentyl(enyl)] heptanoic or heptenoic acids and derivatives of said acids, wherein one or more of said hydroxy groups are replaced by an ether group. The compounds of the present invention are potent ocular hypotensives, and are particularly suitable for the management of glaucoma.

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