Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-09-27
2005-09-27
Seaman, D. Margaret (Department: 1625)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C546S340000, C546S342000, C546S344000, C514S277000
Reexamination Certificate
active
06949656
ABSTRACT:
A composition for use as an antiobestic agent and preventive or therapeutic agent for diabetes, containing a compound of the formula (I):wherein, A is substituted aryl or substituted heteroaryl with one or more group(s); (here, one of following groups is at least contained as the substituent: —RA—RB(RAis S, SO, SO2, NRC, NRCSO2(RCis hydrogen or lower alkyl) or lower alkylene); RBis optionally substituted aryl);X is O, S, NR wherein R is hydrogen or lower alkyl, or single bond;m is an integer of 0 to 4;n is an integer of 1 to 6p is an integer of 1 to 3,pharmaceutically acceptable salt, prodrug or hydrate thereof.
REFERENCES:
patent: 4267183 (1981-05-01), Johnson et al.
patent: 4521428 (1985-06-01), Nisato et al.
patent: 4645771 (1987-02-01), Mills
patent: 6433165 (2002-08-01), Luly et al.
patent: 6649623 (2003-11-01), Yano et al.
patent: 978512 (2000-02-01), None
patent: 2 045 750 (1980-11-01), None
patent: 99/48888 (1999-09-01), None
patent: 00/46194 (2000-08-01), None
DeSantis, Jr., et al., “Synthesis of potential mescaline antagonists”, Journal of Pharmaceutical Sciences, 65(10), pp. 1479-1484 (1976).
Möhrle et al., “Sodium mercury EDTA dehydrogenation of N-aliphatic-substituted 1, 2, 3, 6-tetrahydropyridine derivatives”, Arch. Pharm. (Weinheim), 323(2), pp. 109-115 (1990).
Flann et al., “Iminium ion and acyliminium ion initiated cyclization reactions of vinylsilanes. Regiocontrolled synthesis of tetrahydropyridines and related heterocycles”, J. Am. Chem. Soc., 109(20), pp. 6097-6107 (1987).
Takemura et al., “Synthesis and selective activity of cholinergic agents with rigid skeletons. III”, Chem. Pharm. Bull., 29(10), pp. 3026-3032 (1981).
Ding et al., “A facile synthesis of 3-pyrrolines”, Synthetic Communications, 20(2), pp. 227-230 (1990).
Chapman et al., Polycyclic systems related to [1]benzothieno [2,3-c]pyridine, J. Chem. Soc. (C), (16), pp. 2269-2272 (1970).
Katsuura Goro
Sakaguchi Isako
Yano Toshisada
Yoshikawa Naoki
Seaman D. Margaret
Shionogi & Co. Ltd.
Wenderoth , Lind & Ponack, L.L.P.
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