Cyclic amine derivatives and use thereof

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C546S340000, C546S342000, C546S344000, C514S277000

Reexamination Certificate

active

06949656

ABSTRACT:
A composition for use as an antiobestic agent and preventive or therapeutic agent for diabetes, containing a compound of the formula (I):wherein, A is substituted aryl or substituted heteroaryl with one or more group(s); (here, one of following groups is at least contained as the substituent: —RA—RB(RAis S, SO, SO2, NRC, NRCSO2(RCis hydrogen or lower alkyl) or lower alkylene); RBis optionally substituted aryl);X is O, S, NR wherein R is hydrogen or lower alkyl, or single bond;m is an integer of 0 to 4;n is an integer of 1 to 6p is an integer of 1 to 3,pharmaceutically acceptable salt, prodrug or hydrate thereof.

REFERENCES:
patent: 4267183 (1981-05-01), Johnson et al.
patent: 4521428 (1985-06-01), Nisato et al.
patent: 4645771 (1987-02-01), Mills
patent: 6433165 (2002-08-01), Luly et al.
patent: 6649623 (2003-11-01), Yano et al.
patent: 978512 (2000-02-01), None
patent: 2 045 750 (1980-11-01), None
patent: 99/48888 (1999-09-01), None
patent: 00/46194 (2000-08-01), None
DeSantis, Jr., et al., “Synthesis of potential mescaline antagonists”, Journal of Pharmaceutical Sciences, 65(10), pp. 1479-1484 (1976).
Möhrle et al., “Sodium mercury EDTA dehydrogenation of N-aliphatic-substituted 1, 2, 3, 6-tetrahydropyridine derivatives”, Arch. Pharm. (Weinheim), 323(2), pp. 109-115 (1990).
Flann et al., “Iminium ion and acyliminium ion initiated cyclization reactions of vinylsilanes. Regiocontrolled synthesis of tetrahydropyridines and related heterocycles”, J. Am. Chem. Soc., 109(20), pp. 6097-6107 (1987).
Takemura et al., “Synthesis and selective activity of cholinergic agents with rigid skeletons. III”, Chem. Pharm. Bull., 29(10), pp. 3026-3032 (1981).
Ding et al., “A facile synthesis of 3-pyrrolines”, Synthetic Communications, 20(2), pp. 227-230 (1990).
Chapman et al., Polycyclic systems related to [1]benzothieno [2,3-c]pyridine, J. Chem. Soc. (C), (16), pp. 2269-2272 (1970).

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Cyclic amine derivatives and use thereof does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Cyclic amine derivatives and use thereof, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Cyclic amine derivatives and use thereof will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-3406877

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.