Crystalline isoxazole derivative and medical preparation...

Details Crystalline isoxazole derivative and medical preparation... Crystalline isoxazole derivative and medical preparation...

2002-03-26

2008-09-30

Anderson, Rebecca L (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C544S137000

Reexamination Certificate

active

07429588

ABSTRACT:
Crystalline 3-[(1S)-1-(2-fluorobiphenyl-4-yl)ethyl]-5-{[amino(morpholin-4-yl)methylene]amino}-isoxazole that exhibits the following angle of diffraction (2θ) and relative intensity in a powder X-ray diffraction pattern, is very easy to handle and stable in a process of its formulation into a pharmaceutical preparation.2θ (°)Relative intensity (%)6.110014.15516.07418.53620.04325.439

REFERENCES:
patent: 6100260 (2000-08-01), Nakatsuka et al.
patent: 2005/0158371 (2005-07-01), Nishikado et al.
patent: 1 138 674 (2001-10-01), None
patent: 2000-186038 (2000-07-01), None
patent: 2000-186077 (2000-07-01), None
patent: WO 98/47880 (1998-10-01), None
patent: WO 00/29383 (2000-05-01), None
Brittain polymorphism in pharmaceutical solids Marcel Dekker, p. 1, 2, 178-179, 185, 219 and 236 (1000).
US Pharmacopia #23, national formulary #18, p. 1843-1844, 1995.
A. Maureen Rouhi, Chemical & Engineering News, Feb. 24, 2003, pp. 32-35.
(http://www.ninds.nih.gov/health—and—medical/disorders/aids.htm). accessed May 31, 2004.
Byrn et al. “Solid-State Chemistry of Drugs” (1999), pp. 62-63.
Edited by Sadasuke Okano, Shin•Yakuzaigaku Soron (3rdrevised edition), Kabushiki Kaisha Nankodo, 1987nen, pp. 138, 255, 256.

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