Convergent process for the preparation of a morpholine compound

Details Convergent process for the preparation of a morpholine compound Convergent process for the preparation of a morpholine compound

1999-10-28

2000-04-18

Powers, Fiona T.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

544132, C07D41306, C07D24904

Patent

active

060517174

ABSTRACT:
The present invention is directed to the compound 4-N,N-dimethylaminomethyl-5-formyl-1,2,3-triazole which is a valuable intermediate in the preparation of phamaceutical compounds. The present invention is further directed to a novel convergent process for the preparation of 2-(R)-(1-(R)-(3,5-bis(trifluoromethyl)phenyl)-ethoxy)-4-(5-(dimethylamino) methyl-1,2,3-triazol-4-yl)methyl-3-(S)-(4-fluorophenyl)-morpholine which is a potent and selective substance P (or neurokinin-1) receptor antagonist useful as a therapeutic agent.

REFERENCES:
patent: 5612337 (1997-03-01), Baker et al.

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