Conjugates of biologically active compounds, methods for...

Details Conjugates of biologically active compounds, methods for... Conjugates of biologically active compounds, methods for...

2003-02-14

2009-08-25

McIntosh, III, Traviss C (Department: 1623)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

C514S183000, C536S007100, C536S007200, C536S007400

Reexamination Certificate

active

07579324

ABSTRACT:
This invention features a compound of the following formula:in-line-formulae description="In-line Formulae" end="lead"?T-(-L-C)m,in-line-formulae description="In-line Formulae" end="tail"?T is a transportophore, L is a bond or a linker having a molecular weight up to 240 dalton, C is a non-antibiotic therapeutic agent, and m is 1, 2, 3, 4, 5, 6, 7, or 8, in which the transportophore has an immune selectivity ratio of at least 2, the transportophore is covalently bonded to the non-antibiotic therapeutic agent via the bond or the linker, and the compound has an immune selectivity ratio of at least 2.

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