Conformationally constrained analogs useful as antidiabetic...

Details Conformationally constrained analogs useful as antidiabetic... Conformationally constrained analogs useful as antidiabetic...

2006-09-12

2006-09-12

Coleman, Brenda (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S089000, C514S091000, C514S092000, C514S093000, C514S094000, C514S217030, C514S217040, C514S217080, C514S217090, C514S318000, C514S326000, C514S333000, C514S340000, C514S341000, C514S342000, C514S343000, C514S360000, C514S361000, C514S362000, C514S363000, C514S364000, C514S365000, C514S369000, C514S372000, C514S376000, C514S378000, C514S380000, C514S381000, C514S397000, C514S406000, C514S407000, C514S422000, C514S423000, C514S428000, C540S596000, C540S597000, C540S602000, C540S603000, C546S022000, C546S

Reexamination Certificate

active

07105556

ABSTRACT:
Compounds are provided which have the structurewherein Q is C or N, X1is C or N, and R1, R2, R2a, R2b, R2c, R3, Y, A, m, n, X2, X3and X4are as defined herein, which compounds are useful as antidiabetic, hypolipidemic, and antiobesity agents.

REFERENCES:
patent: 2 027 025 (1979-07-01), None
patent: WO 93/01167 (1992-03-01), None
patent: WO 01/38325 (2000-11-01), None
patent: WO 01/21602 (2001-03-01), None
Davis, Franklin A., et al., Organic Letters, 2001, vol. 3, No. 5, 759-762.
Swarbrick, Martin E., J. Org. Chem. 1999, 64, 1993-2002.
Jeff E. Cobb, et al., “N-(2-Benzoylphenyl)-L-tyrosine PPARy Agonist 3 Structure-Activity Relationship and Optimization of the N-Aryl Substituent”, J. Med. Chem., 1998, 41, 5055-5069.

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