Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-11-08
2010-11-02
Sullivan, Daniel M (Department: 1621)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C549S228000, C549S263000, C549S346000, C549S347000, C549S356000
Reexamination Certificate
active
07825265
ABSTRACT:
Disclosed herein are novel di-aromatic compounds and methods for using various di-aromatic compounds for treatment and prevention of diseases and disorders related to estrogen receptors.
REFERENCES:
patent: 2342294 (1944-02-01), Niederl et al.
patent: 3517071 (1970-06-01), Caldwell et al.
patent: 3829462 (1974-08-01), Krimm et al.
patent: 3872105 (1975-03-01), Grisar et al.
patent: 4082913 (1978-04-01), Suzuki et al.
patent: 4247484 (1981-01-01), Mark et al.
patent: 4554309 (1985-11-01), Mark et al.
patent: 5283374 (1994-02-01), Jeffries et al.
patent: 5691351 (1997-11-01), Kolasa et al.
patent: 6043279 (2000-03-01), Boehm et al.
patent: 6150362 (2000-11-01), Henkin et al.
patent: 6255439 (2001-07-01), Avadhani et al.
patent: 6265402 (2001-07-01), Ina et al.
patent: 6518306 (2003-02-01), Christensen et al.
patent: 6586431 (2003-07-01), Liras et al.
patent: 2005/0256210 (2005-11-01), Olsson et al.
patent: 627224 (1963-07-01), None
patent: 0995737 (2000-04-01), None
patent: 1410275 (1975-10-01), None
patent: 2000-72695 (2000-03-01), None
patent: 00/10958 (2000-02-01), None
patent: WO 00/39091 (2000-07-01), None
patent: 01/10385 (2001-02-01), None
patent: 02/18334 (2002-03-01), None
patent: 2004/048309 (2004-06-01), None
patent: 2005/037755 (2005-04-01), None
Aeberli et al. Journal of Medicinal Chemistry 1969, 12(1), pp. 51-54.
McElvain et al. Journal of the American Chemical Society, 1955, 77, pp. 2848-2850.
Uehara et al. Journal of Organic Chemistry 1999, 64, pp. 1436-1441.
Coleman, K.P. et al., “QSAR Models of the In Vitro Strogen Activity of Bisphenol A Analogs” QSAR Comb. Sci., 2003, 22:78-88.
Database Beilstein, Accession Nos. 3156998, 3519057, 3156998, and 3519057.
Database Beilstein, Accession Nos. 8372608, 9453634, 9455728, 8372608, and 9455728.
Gallegos Saliner, A. et al., “Molecular Quantum Similarity Analysis of Estrogenic Activity”J. Chem. Inf. Comput. Sci., 2003, 43:1166-1176.
Muthyala, R.S. et al., “Bridged Bicyclic Cores Containing a 1,1-Diarylethylene Motif are High-Affinity Subtype-Selective Ligands for the Estrogen Receptor” J. Med. Chem., 2003, 46:1589-1602.
Muthyala, R.S. et al., “Exploration of the Bicyclo[3.3.1]nonane System as a Template for New Ligands for the Estrogen Receptor” Bioorganic & Medicinal Chemistry Letters, 2003, 13:4485-4488.
Niederl, J.B. et al., “Steric Hindrance in Ketone-Phenol Condensations. The Condensation of Guaiacol with Cyclic Ketones” J. Am. Chem. Soc., 1940, 62:320-322.
Yamasaki, K. et al., “Compariosn of the Reporter Gene Assay for ER-alpha Antagonists with the Immature Rat Uterotrophic Assay of 10 Chemicals” Toxicology Letters, 2003, 142:119-131.
Yamasaki, K. et al., “Comparative Study of the Uterotrophic Potency of 14 Chemicals in a Uterotrophic Assay and Their Receptor-Binding Affinity” Toxicology Letters, 2004, 146:111-120.
Office Action, Dated Oct. 29, 2007, U.S. Appl. No. 11/120,397.
Gustafsson Magnus
Hyldtoft Lene
Lund Birgitte Winther
Olsson Roger
Piu Fabrice
ACADIA Pharmaceuticals Inc.
Sullivan Daniel M
Tahmassebi Sam K
TechLaw LLP
Valenrod Yevegeny
LandOfFree
Compounds with activity at estrogen receptors does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Compounds with activity at estrogen receptors, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Compounds with activity at estrogen receptors will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-4201691