Compounds useful as photodynamic therapeutic agents

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Boron containing doai

Reexamination Certificate

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C544S216000, C514S246000

Reexamination Certificate

active

10508754

ABSTRACT:
The present invention relates to compounds of the formulaor a salt, metal complex or hydrate or other solvate thereof, wherein:M is a chelating agent;R1, R2, R3, R4, R5and R6are independently selected from the group consisting of: H; a substituted or unsubstituted, saturated or unsaturated, cyclic, moiety; a substituted or unsubstituted, saturated or unsaturated, heterocyclic moiety; or a substituted or unsubstituted, saturated or unsaturated, straight or branched chain alkyl or acyl moiety; andR2and R5may also be independently a heavy atom or a water-solubilizing group.The present invention also relates to use of these compounds in the therapy in vivo or in vitro of a photosensitive target biological cell by irradiation, as well as methods of treating a photosensitive target biological cell in vivo or in vitro. Finally, the present invention relates to pharmaceutical compositions, comprising these compounds, in association with a pharmaceutically acceptable diluent or carrier.

REFERENCES:
patent: 4916711 (1990-04-01), Boyer et al.
patent: 5326692 (1994-07-01), Brinkley et al.
patent: 5446157 (1995-08-01), Morgan et al.
patent: 361936 (1990-04-01), None
patent: 1253151 (2002-10-01), None
patent: 11092479 (1999-04-01), None
patent: 11092479 (1999-04-01), None
patent: 2000019738 (2000-01-01), None
Takuma, H., Patent Abstracts of Japan, Publication No. 11092479 (Jun. 4, 1999) (Cited in Applicants IDS).
Sathyamoorthi, G., Heteroatom Chemistry, vol. 4(6), pp. 603-608 (1993).
Database Caplus ′Online! Chemical Abstracts Service, Columbus, Ohio, US; 1980, A. Abeysekera et al., “Dicarbonylrhodium(I) complexes of polypyrrole macrocycles. Part 3. Synthesis and crystal structures of complexes of N-methylcorrles, N-methylporphyrins and acyclic polypyrroles”.
J. Killoran et al: “Synthesis of BF2 and chelates of tetraarylazadipyrromethenes and evidence for their photodynamic therapeutic behaviour”, Chem. Comm., vol. 8, No. 17, Aug. 21, 2002, pp. 1862-1863, XP002249180.
International Search Report for International Application No. PCT/EP03/03174.

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