Compounds for the modulation of PPARγ activity

Details Compounds for the modulation of PPARγ activity Compounds for the modulation of PPARγ activity

2004-03-25

2009-12-01

Seaman, D. Margaret (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C546S295000

Reexamination Certificate

active

07626033

ABSTRACT:
Modulators of PPARγ activity are provided which are useful in pharmaceutical compositions and methods for the treatment of conditions such as type II diabetes and obesity.

REFERENCES:
patent: 2407309 (1946-09-01), Lott et al.
patent: 3033870 (1962-05-01), Druey et al.
patent: 3034955 (1962-05-01), Frick et al.
patent: 3174901 (1965-03-01), Sterne
patent: 3669966 (1972-06-01), Ambrogi et al.
patent: 3674843 (1972-07-01), Shen et al.
patent: 3686192 (1972-08-01), Moore et al.
patent: 4003734 (1977-01-01), Johnston
patent: 4013621 (1977-03-01), Knell
patent: 4061642 (1977-12-01), Fleckenstein et al.
patent: 4062950 (1977-12-01), Frommer et al.
patent: 4218237 (1980-08-01), Nishiyama et al.
patent: 4248619 (1981-02-01), Serban et al.
patent: 4289876 (1981-09-01), Algieri et al.
patent: 4499304 (1985-02-01), Gabrielsen et al.
patent: 4549901 (1985-10-01), James
patent: 4565568 (1986-01-01), Johnston et al.
patent: 4572912 (1986-02-01), Yoshioka et al.
patent: 4577028 (1986-03-01), Martin et al.
patent: 4670045 (1987-06-01), Ehr et al.
patent: 4731090 (1988-03-01), Boger et al.
patent: 4756739 (1988-07-01), Fuss et al.
patent: 4851419 (1989-07-01), Cox
patent: 4866079 (1989-09-01), Boger et al.
patent: 4900751 (1990-02-01), Cox
patent: 4946854 (1990-08-01), Maienfisch et al.
patent: 4952235 (1990-08-01), Andree et al.
patent: 4987141 (1991-01-01), Bushell et al.
patent: 5008276 (1991-04-01), Clough et al.
patent: 5070096 (1991-12-01), Mohrs et al.
patent: 5081125 (1992-01-01), Maienfisch et al.
patent: 5093340 (1992-03-01), Mohrs et al.
patent: 5143937 (1992-09-01), Lang et al.
patent: 5151428 (1992-09-01), Sakamoto et al.
patent: 5202336 (1993-04-01), Mohrs et al.
patent: 5204354 (1993-04-01), Chakravarty et al.
patent: 5250549 (1993-10-01), Yoshino et al.
patent: 5304532 (1994-04-01), Munro et al.
patent: 5360810 (1994-11-01), Hayase et al.
patent: 5444036 (1995-08-01), Iwasaki et al.
patent: 5514696 (1996-05-01), Murugesan et al.
patent: 5545669 (1996-08-01), Adams et al.
patent: 5610320 (1997-03-01), Yoshino et al.
patent: 5624937 (1997-04-01), Reel
patent: 5643914 (1997-07-01), Daines
patent: 5684195 (1997-11-01), Huang et al.
patent: 5716993 (1998-02-01), Ozaki et al.
patent: 5780483 (1998-07-01), Widdowson et al.
patent: 5814646 (1998-09-01), Heinz
patent: 5880136 (1999-03-01), Duggan et al.
patent: 5990126 (1999-11-01), Park et al.
patent: 6022897 (2000-02-01), Evans et al.
patent: 6028052 (2000-02-01), Heyman et al.
patent: 6200995 (2001-03-01), De la Brouse-Elwood
patent: 6214850 (2001-04-01), Evans et al.
patent: 6262112 (2001-07-01), Mittendorf et al.
patent: 6294559 (2001-09-01), Smith
patent: 6348474 (2002-02-01), Kayakiri et al.
patent: 6353011 (2002-03-01), Pershadsingh et al.
patent: 6369075 (2002-04-01), Ruggeri et al.
patent: 6376512 (2002-04-01), Jayyosi et al.
patent: 6403607 (2002-06-01), Hidaka et al.
patent: 6469054 (2002-10-01), Mittendorf et al.
patent: 6472779 (2002-10-01), Hwang et al.
patent: 6545050 (2003-04-01), Mittendorf et al.
patent: 6573278 (2003-06-01), Mittendorf et al.
patent: 6583157 (2003-06-01), McGee et al.
patent: 6586475 (2003-07-01), Kato et al.
patent: 6620827 (2003-09-01), De la Brouse-Elwood et al.
patent: 6653309 (2003-11-01), Saunders et al.
patent: 6653332 (2003-11-01), Jaen et al.
patent: 6770648 (2004-08-01), McGee et al.
patent: 7041691 (2006-05-01), McGee et al.
patent: 7132546 (2006-11-01), Kato et al.
patent: 7223761 (2007-05-01), Kruk et al.
patent: 7439242 (2008-10-01), Houze et al.
patent: 2001/0028200 (2001-10-01), Hwang et al.
patent: 2003/0088103 (2003-05-01), Houze et al.
patent: 2003/0171399 (2003-09-01), McGee et al.
patent: 2004/0048891 (2004-03-01), Kato et al.
patent: 2004/0176409 (2004-09-01), McGee et al.
patent: 592 411 (1977-10-01), None
patent: 3632329 (1988-03-01), None
patent: 0 069 585 (1983-01-01), None
patent: 0 148 730 (1985-07-01), None
patent: 0 261 539 (1987-09-01), None
patent: 0 261 539 (1988-03-01), None
patent: 0 306 222 (1989-03-01), None
patent: 0 778 267 (1996-11-01), None
patent: 0 749 751 (1996-12-01), None
patent: 0 472 053 (1998-06-01), None
patent: 0 855 391 (1998-07-01), None
patent: 2373725 (2002-10-01), None
patent: 55-79369 (1980-06-01), None
patent: 64-6245 (1989-01-01), None
patent: 9-255656 (1997-09-01), None
patent: WO 95/01326 (1995-01-01), None
patent: WO 95/33461 (1995-12-01), None
patent: WO 95/33462 (1995-12-01), None
patent: WO 96/09294 (1996-03-01), None
patent: WO 96/15118 (1996-05-01), None
patent: WO 97/00857 (1997-01-01), None
patent: WO 97/30677 (1997-08-01), None
patent: WO 97/31907 (1997-09-01), None
patent: WO 97/36579 (1997-10-01), None
patent: WO 98/02437 (1998-01-01), None
patent: WO 98/16503 (1998-04-01), None
patent: WO 98/27081 (1998-06-01), None
patent: WO 98/37061 (1998-08-01), None
patent: WO 98/50029 (1998-11-01), None
patent: WO 98/50030 (1998-11-01), None
patent: WO 98/50030 (1998-11-01), None
patent: WO 99/00372 (1999-01-01), None
patent: WO 99/06378 (1999-02-01), None
patent: WO 99/10320 (1999-03-01), None
patent: WO 99/20275 (1999-04-01), None
patent: WO 99/24404 (1999-05-01), None
patent: WO 99/32465 (1999-07-01), None
patent: WO 99/38845 (1999-08-01), None
patent: WO 99/50237 (1999-10-01), None
patent: WO 99/55663 (1999-11-01), None
patent: WO 00/10967 (2000-03-01), None
patent: WO 00/10968 (2000-03-01), None
patent: WO 00/12073 (2000-03-01), None
patent: WO 00/12623 (2000-03-01), None
patent: WO 00/17202 (2000-03-01), None
patent: WO 00/31021 (2000-06-01), None
patent: WO 01/00579 (2001-01-01), None
patent: WO 01/30343 (2001-05-01), None
patent: WO 01/60807 (2001-08-01), None
patent: WO 01/70723 (2001-09-01), None
patent: WO 01/82916 (2001-11-01), None
patent: WO 01/83427 (2001-11-01), None
patent: WO 01/87861 (2001-11-01), None
patent: WO 01/95906 (2001-12-01), None
patent: WO 02/00611 (2002-01-01), None
patent: WO 02/08188 (2002-01-01), None
patent: WO 02/13812 (2002-02-01), None
patent: WO 02/13864 (2002-02-01), None
patent: WO 02/14291 (2002-02-01), None
patent: WO 02/17901 (2002-03-01), None
patent: WO 02/18355 (2002-03-01), None
patent: WO 02/26729 (2002-04-01), None
patent: WO 02/26737 (2002-04-01), None
patent: WO 02/28832 (2002-04-01), None
patent: WO 02/28857 (2002-04-01), None
patent: WO 02/30860 (2002-04-01), None
patent: WO 02/30863 (2002-04-01), None
patent: WO 02/30884 (2002-04-01), None
patent: WO 02/30895 (2002-04-01), None
patent: WO 02/40020 (2002-05-01), None
patent: WO 02/46161 (2002-06-01), None
patent: WO 02/49626 (2002-06-01), None
patent: WO 02/051397 (2002-07-01), None
patent: WO 02/051820 (2002-07-01), None
patent: WO 02/053546 (2002-07-01), None
patent: WO 02/059098 (2002-08-01), None
patent: WO 02/060434 (2002-08-01), None
patent: WO 02/062772 (2002-08-01), None
patent: WO 02/062774 (2002-08-01), None
patent: WO 02/062798 (2002-08-01), None
patent: WO 02/062799 (2002-08-01), None
patent: WO 02/064094 (2002-08-01), None
patent: WO 02/066028 (2002-08-01), None
patent: WO 02/072003 (2002-09-01), None
patent: WO 02/074291 (2002-09-01), None
patent: WO 02/080913 (2002-10-01), None
patent: WO 02/081454 (2002-10-01), None
patent: WO 01/87860 (2002-11-01), None
patent: WO 01/87862 (2002-11-01), None
patent: WO 02/092084 (2002-11-01), None
patent: WO 02/092590 (2002-11-01), None
U.S. Appl. No. 09/606,433, filed Jun. 28, 2000, McGee et al.
U.S. Appl. No. 10/719,997, filed Nov. 20, 2003, McGee et al.
Willson et al., “The PPARs: from orphan receptors to drug discovery” J. Med. Chem. 43(4):527-550 (2000).
U.S. Appl. No. 10/456,932, filed Jun. 5, 2003, Jaen et al.
Badilescu, I., “Sythesis of some N-aryl- and N,N-dialkyl-p-chloro-benzensulfonamides” Rev.Chim., vol. 17, No. 11, 1966, pp. 705-706 & Chemical Abstracts, vol. 67, No. 9, Aug. 28, 1967, Columbus, Ohio, United States; abstract No. 43516y, p. 4076; XP002099084.
Baguley et al., Database accession No. 108:179602, Database Chemabs ′Online!, RN 106831-10-1 CAPLUS, Eur. J. Cancer Clin. Oncol., 24(2):205-210 (1988).
Burmistrov et al., Database accession No. 115:8165, Database Chemabs ′Online!, RNs 98187-76-9 CAPLUS, 134284-40-5 C

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