Compounds and medicinal use thereof

Details Compounds and medicinal use thereof Compounds and medicinal use thereof

2008-01-01

2008-01-01

O'Sullivan, Peter (Department: 1621)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Ester doai

C514S538000, C514S539000, C514S544000, C514S545000, C514S567000, C514S568000, C514S570000, C514S571000, C560S009000, C560S019000, C560S020000, C560S021000, C560S052000, C560S101000, C562S426000, C562S435000, C562S441000, C562S560000

Reexamination Certificate

active

09830559

ABSTRACT:
A compound or a salt thereof having the atom corresponding to N3and the two or more atoms selected from N1, N2, N4and N5, said atoms constitute the pharmacophore represented by the following formula:and inhibits the activity of transcription factor AP-1 and is useful as an agent for preventing and treating the diseases into which over expression of AP-1 participates and as an AP-1 inhibitor.

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