Drug – bio-affecting and body treating compositions – Preparations characterized by special physical form – Particulate form
Patent
1998-09-03
2000-10-10
Rose, Shep K.
Drug, bio-affecting and body treating compositions
Preparations characterized by special physical form
Particulate form
424465, A61K 916, A61K 920
Patent
active
061299324
ABSTRACT:
The invention is a pharmaceutical composition for oral administration to a patient comprising pharmaceutically effective amount of [3(R)-[2-Piperidin-4-yl)ethyl]-2-piperidone-1]acetyl-3(R)-methyl-.beta.-al anine, or a pharmaceutically acceptable salt thereof; pharmaceutically acceptable amounts of a polymeric binder; and pharmaceutically acceptable amounts of pharmaceutically acceptable excipients.
The invention is also a process for making a pharmaceutical composition comprising [3(R)-[2-Piperidin-4-yl)ethyl]-2-piperidone-1]acetyl-3(R)-methyl-.beta.-al anine, which comprises the steps of
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Asgharnejad Mandana
Shiromani Prafull K.
Merck & Co. , Inc.
Parr Richard S.
Rose Shep K.
Winokur Melvin
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