Compositions comprising 1-substituted azacycloalkanes

Details Compositions comprising 1-substituted azacycloalkanes Compositions comprising 1-substituted azacycloalkanes

1990-11-13

1993-10-26

Ore, Dale R.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

8405, 8406, 424DIG5, 424DIG10, 424DIG13, 424 47, 424 59, 424 60, 424 61, 424 63, 424 70, 514 29, 514192, 5142235, 514844, 514846, 514858, 514859, 514861, 514862, 514863, 514864, 514880, 514881, 514885, 514886, 514887, 514912, 514918, 514944, 514946, 514947, 514965, 514969, 523297, 536 165, A01N 4304, A61K 3170, A61K 742, A61K 744, A61K 902, A61K 906, A61K 910, A61K 912

Patent

active

052566471

ABSTRACT:
This invention provides compositions comprising a physiologically-active agent and a compound having the structural formula ##STR1## wherein X may represent sulfur or two hydrogen atoms; R' is H or a lower alkyl group having 1-4 carbon atoms; m is 2-6; n is 0-18 and R is --CH.sub.3, ##STR2## wherein R" is H or halogen, in an amount effective to enhance the penetration of the physiologically-active agent through the skin or other membrane of the body of an animal.

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